Compile Data Set for Download or QSAR
maximum 50k data
Found 21 with Last Name = 'alekshun' and Initial = 'mn'
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50371227(CHEMBL400462)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319090((E)-3-(4-Acetyl-phenyl)-N-[4-(1-hydroxy-6-nitro-1H...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378357(CHEMBL575329)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319080((E)-N-(4-(6-cyano-1-hydroxy-1H-benzo[d]imidazol-2-...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319088((E)-2-(2-(4-(3-(4-acetylphenyl)acrylamido)phenyl)-...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50371226(CHEMBL251209)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319089((E)-2-(2-(4-(3-(6-acetylpyridin-3-yl)acrylamido)ph...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378358(CHEMBL572948)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50378359(CHEMBL575963)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa ExsA binding to DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319081((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319079((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319078((E)-N-(4-(6-cyano-1-hydroxy-1H-benzo[d]imidazol-2-...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319092((E)-3-(6-acetylpyridin-3-yl)-N-(4-(1-hydroxy-6-nit...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319093((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319091((E)-3-(4-acetylphenyl)-N-(4-(6-cyano-1-hydroxy-1H-...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa 388 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319082((E)-3-(6-(1H-imidazol-1-yl)pyridin-3-yl)-N-(4-(1-h...)
Affinity DataIC50:  3.12E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319085((E)-3-(4-acetylphenyl)-N-(2-amino-2-oxoethyl)-N-(4...)
Affinity DataIC50: >4.75E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319086((E)-3-(4-acetylphenyl)-N-(2-amino-2-oxoethyl)-N-(4...)
Affinity DataIC50: >4.90E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319087((E)-2-(3-(4-acetylphenyl)-N-(4-(6-cyano-1-hydroxy-...)
Affinity DataIC50: >5.10E+4nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319083((E)-3-(6-(dimethylamino)pyridin-3-yl)-N-(4-(1-hydr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator ExsA(Pseudomonas aeruginosa)
Paratek Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50319084((E)-N-(4-(1-hydroxy-6-nitro-1H-benzo[d]imidazol-2-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Pseudomonas aeruginosa PAO1 ExsA DNA binding activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed