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Found 100 with Last Name = 'alemayehu' and Initial = 's'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171546((S)-2,4-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  0.480nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  0.720nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171653(CHEMBL196120 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  0.800nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171556((R)-1-((S)-2-amino-3-methylbutanamido)ethylboronic...)
Affinity DataIC50:  0.890nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171648(CHEMBL372180 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171649(CHEMBL196933 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  2nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171645(2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171558(2,6-Diamino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  3.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171650(2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171656(2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  4.10nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171647(CHEMBL373269 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  4.60nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171553(2,5-Diamino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171653(CHEMBL196120 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  6.30nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  6.70nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171649(CHEMBL196933 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  7.80nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171647(CHEMBL373269 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171657(2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171559((S)-2,3-Diamino-N-((R)-1-boron-dihydroxide-pentyl)...)
Affinity DataIC50:  8.20nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against human fibroblast activation protein alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171644(CHEMBL427012 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171651(2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50:  15nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171551((S)-2-Amino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171657(2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171651(2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171650(2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171656(2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  27nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171548((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  30nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171652(CHEMBL381444 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50:  38nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50050517(Boronic acid derivative | CHEMBL305170 | N-alkyl G...)
Affinity DataIC50:  38nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171557((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-3-m...)
Affinity DataIC50:  40nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171547((S)-2-Amino-N-((R)-1-boron-dihydroxide-pentyl)-but...)
Affinity DataIC50:  49nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171645(2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  58nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171648(CHEMBL372180 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  61nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171551((S)-2-Amino-hexanoic acid ((R)-1-boron-dihydroxide...)
Affinity DataIC50:  65nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171550((S)-2-Amino-pentanoic acid ((R)-1-boron-dihydroxid...)
Affinity DataIC50:  71nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171655(2-Cyclobutylamino-1-pyrrolidin-1-yl--2-borandihydr...)
Affinity DataIC50:  75nMAssay Description:Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 8(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171555((S)-2,4-Diamino-1-(2-boron-dihydroxide-pyrrolidin-...)
Affinity DataIC50:  95nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 8 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171644(CHEMBL427012 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  99nMAssay Description:Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171644(CHEMBL427012 | N-alkyl Gly-boro-Pro derivative)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50171561((S)-2,4-Diamino-4-piperidin-1-yl-butyric acid | CH...)
Affinity DataIC50:  130nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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