Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universitat Pompeu Fabra
Curated by ChEMBL
Universitat Pompeu Fabra
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Binding affinity at rat 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universitat Pompeu Fabra
Curated by ChEMBL
Universitat Pompeu Fabra
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Binding affinity at rat 5HT2A receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 137nMAssay Description:Displacement of [3H]-spiperone from cloned human dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 182nMAssay Description:Displacement of [3H]-spiperone from cloned human dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 199nMAssay Description:Displacement of [3H]-spiperone from cloned human dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 212nMAssay Description:Displacement of [3H]-spiperone from cloned human dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 227nMAssay Description:Displacement of [3H]-spiperone from cloned human dopamine D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 228nMAssay Description:Displacement of [3H]-spiperone from cloned human dopamine D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universitat Pompeu Fabra
Curated by ChEMBL
Universitat Pompeu Fabra
Curated by ChEMBL
Affinity DataKi: 275nMAssay Description:Binding affinity at rat 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 458nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 829nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universitat Pompeu Fabra
Curated by ChEMBL
Universitat Pompeu Fabra
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity at rat 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universitat Pompeu Fabra
Curated by ChEMBL
Universitat Pompeu Fabra
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity at rat 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.94E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.08E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.59E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.16E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.69E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universitat Pompeu Fabra
Curated by ChEMBL
Universitat Pompeu Fabra
Curated by ChEMBL
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity at rat 5HT2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universitat Pompeu Fabra
Curated by ChEMBL
Universitat Pompeu Fabra
Curated by ChEMBL
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity at rat 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.82E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.79E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 178nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 467nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 223nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 524nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 183nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: 121nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPre-mRNA-processing factor 19(Saccharomyces cerevisiae S288c)
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Polymer Functionalization Group (Ictp, Csic)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in human MCF7 cells coexpressing TIF2 by luciferase reporter gene assayMore data for this Ligand-Target Pair