TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Kumamoto University
Curated by ChEMBL
Kumamoto University
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of [3H]-farnesyl pyrophosphate binding to human farnesyltransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Kumamoto University
Curated by ChEMBL
Kumamoto University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of [3H]-farnesyl pyrophosphate binding to human farnesyltransferaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 2.65E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.07E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.64E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 4.03E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 4.94E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Kumamoto University
Curated by ChEMBL
Kumamoto University
Curated by ChEMBL
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of [3H]-farnesyl pyrophosphate binding to human farnesyltransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Kumamoto University
Curated by ChEMBL
Kumamoto University
Curated by ChEMBL
Affinity DataIC50: 6.20E+5nMAssay Description:Inhibition of [3H]-farnesyl pyrophosphate binding to human farnesyltransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Kumamoto University
Curated by ChEMBL
Kumamoto University
Curated by ChEMBL
Affinity DataIC50: 4.00E+6nMAssay Description:Inhibition of [3H]-farnesyl pyrophosphate binding to human farnesyltransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Kumamoto University
Curated by ChEMBL
Kumamoto University
Curated by ChEMBL
Affinity DataIC50: 1.55E+7nMAssay Description:Inhibition of [3H]-farnesyl pyrophosphate binding to human farnesyltransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Kumamoto University
Curated by ChEMBL
Kumamoto University
Curated by ChEMBL
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibition of [3H]-farnesyl pyrophosphate binding to human farnesyltransferaseMore data for this Ligand-Target Pair