Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of human COX2 expressed in insect cells using arachidonic acid as substrate pretreated for 3 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.46E+4nMAssay Description:Inhibition of human COX2 expressed in insect cells using arachidonic acid as substrate pretreated for 3 mins followed by substrate addition measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.68E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate pretreated for 3 mins followed by substrate addition measured immediatelyMore data for this Ligand-Target Pair
Affinity DataIC50: 4.53E+4nMAssay Description:Inhibition of type-2 human steroid 5-alpha-reductase.More data for this Ligand-Target Pair
Affinity DataIC50: 4.77E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate pretreated for 3 mins followed by substrate addition measured immediatelyMore data for this Ligand-Target Pair
Affinity DataIC50: 5.22E+4nMAssay Description:Inhibitory concentration required for in vitro binding affinity to cholinergic central Nicotinic acetylcholine receptor on rat brain cortex by using ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.22E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate pretreated for 3 mins followed by substrate addition measured immediatelyMore data for this Ligand-Target Pair
Affinity DataIC50: 5.25E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate pretreated for 3 mins followed by substrate addition measured immediatelyMore data for this Ligand-Target Pair
Affinity DataIC50: 5.64E+4nMAssay Description:Antagonistic potency for NK-1 receptor was determined in vitro,using isolated rabbit vena cava.More data for this Ligand-Target Pair
Affinity DataIC50: 7.28E+4nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate pretreated for 3 mins followed by substrate addition measured immediatelyMore data for this Ligand-Target Pair
Affinity DataIC50: 8.11E+4nMAssay Description:Antagonistic potency for NK-3 receptor was determined in vitro using isolated rat portal vein.More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+5nMAssay Description:Antagonistic potency for NK-1 receptor was determined in a radioligand binding assay using IM9 human lymphoblastoma cell line.More data for this Ligand-Target Pair