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Found 23 with Last Name = 'amici' and Initial = 'md'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50110258((6S)-2-(6-chloropyridin-3-yl)-9-azabicyclo[4.2.1]n...)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]epibatidine from nAChR alpha4beta2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50110258((6S)-2-(6-chloropyridin-3-yl)-9-azabicyclo[4.2.1]n...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]nicotine from nAChR alpha4beta2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50135594((+/-)-2-(6-chloropyridin-3-yl)-9-aza-bicyclo[4.2.1...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]methyllycaconitine from nAChR alpha7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50291551(CHEMBL274329 | Trimethyl-[4-(3-oxo-isoxazolidin-2-...)
Affinity DataIC50:  0.800nMAssay Description:Muscarinic receptor M2 in rat heart using [3H]-QNB (quinuclidinyl benzylate) radioligand as a M2 non-selective muscarinic receptor antagonist at a co...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50223182(2-(4-(pyrrolidin-1-yl)but-2-ynyl)isoxazolidin-3-on...)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataIC50:  2nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291550(3-(4-Pyrrolidin-1-yl-but-2-ynyloxy)-4,5-dihydro-is...)
Affinity DataIC50:  4nMAssay Description:Compound was assessed for the binding affinity against muscarinic receptor subtypes in rat brain using [3H]OXO-M radioligand as a muscarinic receptor...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291552(2-(4-Dimethylamino-but-2-ynyl)-isoxazolidin-3-one ...)
Affinity DataIC50:  23nMAssay Description:Compound was assessed for the binding affinity against muscarinic receptor subtypes in rat brain using [3H]OXO-M radioligand as a muscarinic receptor...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291551(CHEMBL274329 | Trimethyl-[4-(3-oxo-isoxazolidin-2-...)
Affinity DataIC50:  74nMAssay Description:Muscarinic receptor M2 in rat heart using [3H]QNB (quinuclidinyl benzylate) radioligand as a M2 non-selective muscarinic receptor antagonist at a con...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50223182(2-(4-(pyrrolidin-1-yl)but-2-ynyl)isoxazolidin-3-on...)
Affinity DataIC50:  78nMAssay Description:Binding affinity against Muscarinic receptor M1 in rat brain using [3H]-PZ (pirenzepine) radioligand at a concentration of 1 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataIC50:  84nMAssay Description:Muscarinic receptor M2 in rat heart using [3H]-QNB (quinuclidinyl benzylate) radioligand as a M2 non-selective muscarinic receptor antagonist at a co...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataIC50:  100nMAssay Description:Binding affinity against Muscarinic receptor M1 in rat brain using [3H]-PZ (pirenzepine) radioligand at a concentration of 1 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50223182(2-(4-(pyrrolidin-1-yl)but-2-ynyl)isoxazolidin-3-on...)
Affinity DataIC50:  215nMAssay Description:Muscarinic receptor M2 in rat heart using [3H]-QNB (quinuclidinyl benzylate) radioligand as a M2 non-selective muscarinic receptor antagonist at a co...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291550(3-(4-Pyrrolidin-1-yl-but-2-ynyloxy)-4,5-dihydro-is...)
Affinity DataIC50:  233nMAssay Description:Muscarinic receptor M2 in rat heart using [3H]-QNB (quinuclidinyl benzylate) radioligand as a M2 non-selective muscarinic receptor antagonist at a co...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291550(3-(4-Pyrrolidin-1-yl-but-2-ynyloxy)-4,5-dihydro-is...)
Affinity DataIC50:  412nMAssay Description:Binding affinity against Muscarinic receptor M1 in rat brain using [3H]-PZ (pirenzepine) radioligand at a concentration of 1 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291551(CHEMBL274329 | Trimethyl-[4-(3-oxo-isoxazolidin-2-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Binding affinity against Muscarinic receptor M1 in rat brain using [3H]-PZ (pirenzepine) radioligand at a concentration of 1 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291552(2-(4-Dimethylamino-but-2-ynyl)-isoxazolidin-3-one ...)
Affinity DataIC50:  1.38E+3nMAssay Description:Muscarinic receptor M2 in rat heart using [3H]-QNB (quinuclidinyl benzylate) radioligand as a M2 non-selective muscarinic receptor antagonist at a co...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataIC50:  2.00E+3nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50223182(2-(4-(pyrrolidin-1-yl)but-2-ynyl)isoxazolidin-3-on...)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291552(2-(4-Dimethylamino-but-2-ynyl)-isoxazolidin-3-one ...)
Affinity DataIC50:  7.10E+3nMAssay Description:Binding affinity against Muscarinic receptor M1 in rat brain using [3H]-PZ (pirenzepine) radioligand at a concentration of 1 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291550(3-(4-Pyrrolidin-1-yl-but-2-ynyloxy)-4,5-dihydro-is...)
Affinity DataIC50:  8.60E+3nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291551(CHEMBL274329 | Trimethyl-[4-(3-oxo-isoxazolidin-2-...)
Affinity DataIC50:  1.74E+4nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50291552(2-(4-Dimethylamino-but-2-ynyl)-isoxazolidin-3-one ...)
Affinity DataIC50:  1.01E+5nMAssay Description:Binding affinity against Muscarinic receptor M2 in rat brain using [3H]-QNB (quinuclidinyl benzylate) radioligand at a concentration of 0.12 nMMore data for this Ligand-Target Pair
In DepthDetails Article