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Found 389 with Last Name = 'amoroso' and Initial = 'r'
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50595010(CHEMBL5196990)
Affinity DataKi:  10nMAssay Description:Binding affinity to carbonic anhydrase 2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50142631(CHEMBL3758997)
Affinity DataKi:  16nMAssay Description:Binding affinity to carbonic anhydrase 2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50595008(CHEMBL5181066)
Affinity DataKi:  16nMAssay Description:Binding affinity to carbonic anhydrase 2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50142631(CHEMBL3758997)
Affinity DataKi:  21nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50595008(CHEMBL5181066)
Affinity DataKi:  21nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50595009(CHEMBL5170213)
Affinity DataKi:  21nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50595008(CHEMBL5181066)
Affinity DataKi:  32nMAssay Description:Binding affinity to carbonic anhydrase 1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50595009(CHEMBL5170213)
Affinity DataKi:  32nMAssay Description:Binding affinity to carbonic anhydrase 1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50142631(CHEMBL3758997)
Affinity DataKi:  32nMAssay Description:Binding affinity to carbonic anhydrase 1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50595010(CHEMBL5196990)
Affinity DataKi:  78nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  94nMAssay Description:Binding affinity to carbonic anhydrase 2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataKi:  110nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  436nMAssay Description:Binding affinity to carbonic anhydrase 1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50142631(CHEMBL3758997)
Affinity DataKi:  2.54E+3nMAssay Description:Binding affinity to AChE (unknown origin) assessed as inhibition constant using AChI as substrate incubated for 15 mins by Ellman's spectrophotometri...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50435764(CHEMBL2392692)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50217448(CHEMBL242459 | US9029401, 1471 (t-AUCB) | trans-4-...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of aromatase in human MCF-7aro cells using [1beta-3H] androstenedione as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataIC50:  2nMAssay Description:Inhibition of AT1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  4nMAssay Description:Inhibition of AChE (unknown origin) incubated for 30 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171310(CHEMBL3805814)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171231(CHEMBL3805851)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171227(CHEMBL3806301)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50345657(CHEMBL1784801 | rac-3-((1H-imidazol-1-yl)methyl)-1...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50543107(CHEMBL4633346)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171229(CHEMBL3805211)
Affinity DataIC50:  13nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171390(CHEMBL3805733)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171226(CHEMBL3805173)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171228(CHEMBL3805481)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171345(CHEMBL3805008)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171348(CHEMBL3806075)
Affinity DataIC50:  21nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171350(CHEMBL3805539)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171208(CHEMBL3805310)
Affinity DataIC50:  24nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171308(CHEMBL3806046)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171311(CHEMBL3805149)
Affinity DataIC50:  42nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171307(CHEMBL3806159)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
"G. D'Annunzio" University Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM10989((1R)-N-(prop-2-yn-1-yl)-2,3-dihydro-1H-inden-1-ami...)
Affinity DataIC50:  44nMAssay Description:Inhibition of MAO-B (unknown origin) incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171346(CHEMBL3805388)
Affinity DataIC50:  45nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171309(CHEMBL3805839)
Affinity DataIC50:  46nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171342(CHEMBL3806185)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171344(CHEMBL3805657)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171312(CHEMBL3805048)
Affinity DataIC50:  51nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171207(CHEMBL3805021)
Affinity DataIC50:  53nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171230(CHEMBL3806151)
Affinity DataIC50:  54nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio

Curated by ChEMBL
LigandPNGBDBM50401339(CHEMBL4161447)
Affinity DataIC50:  58nMAssay Description:Inhibition of recombinant mouse iNOS using [3H]L-arginine as substrate preincubated for 15 mins followed by NADPH addition measured after 20 mins in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171349(CHEMBL3805820)
Affinity DataIC50:  59nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
University Of Chieti "G. D.Annunzio

Curated by ChEMBL
LigandPNGBDBM25737(12-[(adamantan-1-ylcarbamoyl)amino]dodecanoic acid...)
Affinity DataIC50:  69nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50171306(CHEMBL3806282)
Affinity DataIC50:  79nMAssay Description:Inhibition of recombinant human aromatase using 7-methoxy-4-trifluoromethyl coumarin as substrate measured at anoxic conditions by fluorescence analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara

Curated by ChEMBL
LigandPNGBDBM50226527(CHEMBL107251 | N-(3-(AMINOMETHYL)BENZYL)ACETAMIDIN...)
Affinity DataIC50:  80nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
University Of Chieti "G. D'Annunzio

Curated by ChEMBL
LigandPNGBDBM50226527(CHEMBL107251 | N-(3-(AMINOMETHYL)BENZYL)ACETAMIDIN...)
Affinity DataIC50:  100nMAssay Description:Inhibition of mouse recombinant iNOS using [3H]L-arginine substrate assessed as formation of [3H]L-citruline by liquid scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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