Affinity DataKi: 0.398nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.933nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.37nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.01nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.59nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 851nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.513nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.575nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.631nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.759nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.776nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.32nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.48nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.48nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.55nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.82nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.57nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.63nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.37nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.03nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.13nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.32nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.91nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.33nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 11.2nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 11.5nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 13.5nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 22.4nMAssay Description:Antagonist activity against human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Cape Town
Curated by ChEMBL
University Of Cape Town
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Cape Town
Curated by ChEMBL
University Of Cape Town
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+5nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+5nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+5nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+5nMAssay Description:Binding affinity to TTR in human plasma assessed as protein stabilization preincubated for 1 hr followed by urea-mediated denaturation by Western blo...More data for this Ligand-Target Pair