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Found 28 with Last Name = 'anastasio' and Initial = 'mb'
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071250(CHEMBL292545 | [(S)-3-((R)-2-Hydroxycarbamoylmethy...)
Affinity DataIC50:  11nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071248(CHEMBL416857 | {(S)-3-[(R)-2-((R)-1-Hydroxycarbamo...)
Affinity DataIC50:  21nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071246((2R,3R)-N*1*-Hydroxy-N*4*-[(S)-1-(2-methoxy-ethyl)...)
Affinity DataIC50:  30nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071256(CHEMBL417574 | {(S)-3-[(R)-2-((R)-1-Hydroxycarbamo...)
Affinity DataIC50:  49nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071244((2R,3R)-N*1*-Hydroxy-2-(3-hydroxy-propyl)-3-isobut...)
Affinity DataIC50:  51nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071248(CHEMBL416857 | {(S)-3-[(R)-2-((R)-1-Hydroxycarbamo...)
Affinity DataIC50:  57nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071251(CHEMBL62436 | [(S)-3-((2R,3R)-3-Hydroxycarbamoyl-2...)
Affinity DataIC50:  58nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071254((2R,3R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-(2-met...)
Affinity DataIC50:  83nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071254((2R,3R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-1-(2-met...)
Affinity DataIC50:  94nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071251(CHEMBL62436 | [(S)-3-((2R,3R)-3-Hydroxycarbamoyl-2...)
Affinity DataIC50:  96nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071244((2R,3R)-N*1*-Hydroxy-2-(3-hydroxy-propyl)-3-isobut...)
Affinity DataIC50:  104nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071253((2R,3S)-N*1*-Hydroxy-N*4*-[(S)-1-(2-methoxy-ethyl)...)
Affinity DataIC50:  108nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071246((2R,3R)-N*1*-Hydroxy-N*4*-[(S)-1-(2-methoxy-ethyl)...)
Affinity DataIC50:  112nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071247((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-2-oxo-1-(2-p...)
Affinity DataIC50:  117nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071255(CHEMBL61679 | [(S)-3-((R)-2-Hydroxycarbamoylmethyl...)
Affinity DataIC50:  129nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071249((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-2-oxo-1-(3-p...)
Affinity DataIC50:  140nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071256(CHEMBL417574 | {(S)-3-[(R)-2-((R)-1-Hydroxycarbamo...)
Affinity DataIC50:  215nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071245(CHEMBL62709 | [(S)-3-((R)-2-Hydroxycarbamoylmethyl...)
Affinity DataIC50:  225nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071243((R)-N*4*-Hydroxy-N*1*-[(S)-1-(2-methoxy-ethyl)-2-o...)
Affinity DataIC50:  250nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071247((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-2-oxo-1-(2-p...)
Affinity DataIC50:  518nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071255(CHEMBL61679 | [(S)-3-((R)-2-Hydroxycarbamoylmethyl...)
Affinity DataIC50:  824nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071250(CHEMBL292545 | [(S)-3-((R)-2-Hydroxycarbamoylmethy...)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071249((R)-N*4*-Hydroxy-2-isobutyl-N*1*-[(S)-2-oxo-1-(3-p...)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071243((R)-N*4*-Hydroxy-N*1*-[(S)-1-(2-methoxy-ethyl)-2-o...)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071245(CHEMBL62709 | [(S)-3-((R)-2-Hydroxycarbamoylmethyl...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071252((R)-N*4*-Hydroxy-2-isobutyl-N*1*-((S)-2-oxo-azepan...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071253((2R,3S)-N*1*-Hydroxy-N*4*-[(S)-1-(2-methoxy-ethyl)...)
Affinity DataIC50:  4.36E+3nMAssay Description:Inhibition of matrix metalloproteinase-1 (MMP-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071252((R)-N*4*-Hydroxy-2-isobutyl-N*1*-((S)-2-oxo-azepan...)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of matrix metalloproteinase-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed