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Found 139 with Last Name = 'andressen' and Initial = 'kw'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483188(CHEMBL1632166)
Affinity DataKi:  0.00145nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0398nMAssay Description:Displacement of [3H]GR113808 from human 5-HT4B receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483175(CHEMBL1632165)
Affinity DataKi:  0.0427nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023377(CHEMBL3329805)
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.0525nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483174(CHEMBL1632163)
Affinity DataKi:  0.0537nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483187(CHEMBL1632169)
Affinity DataKi:  0.0646nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0741nMAssay Description:Antagonistic activity at human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023365(CHEMBL3329814)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]GR113808 from human 5-HT4B receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483173(CHEMBL1632157)
Affinity DataKi:  0.102nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483172(CHEMBL1632158)
Affinity DataKi:  0.107nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50492064(CHEMBL2391994)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]GR113808 from human 5-HT4B receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483186(CHEMBL1632167)
Affinity DataKi:  0.141nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483171(CHEMBL1632159)
Affinity DataKi:  0.195nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023375(CHEMBL3329807)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023373(CHEMBL3329809)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023379(CHEMBL3329803)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023376(CHEMBL3329806)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483191(CHEMBL1632162)
Affinity DataKi:  0.234nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023374(CHEMBL3329808)
Affinity DataKi:  0.251nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023366(CHEMBL3329813)
Affinity DataKi:  0.316nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483169(CHEMBL1632160)
Affinity DataKi:  0.339nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483170(CHEMBL1632168)
Affinity DataKi:  0.339nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483182(CHEMBL1632161)
Affinity DataKi:  0.759nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50442803(CHEMBL2440453)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]SB207710 from 5-HT4 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483178(CHEMBL1632154)
Affinity DataKi:  0.813nMAssay Description:Antagonistic activity at human 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023378(CHEMBL3329804)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483184(CHEMBL1632171)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023368(CHEMBL3329812)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023372(CHEMBL3329810)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023367(CHEMBL3329811)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483181(CHEMBL1632164)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50009298(CHEMBL3233521)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]Triptorelin from rat full-length gonadotropin-releasing hormone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483176(CHEMBL1632174)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50023369(CHEMBL3329226)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]GR113808 from human 5HT4b receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM85026(N-(1-Butylpiperidine-4-ylmethyl)-1,2-(trimethylene...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]SB207710 from 5-HT4 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483183(CHEMBL1632172)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483180(CHEMBL1632173)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Mus musculus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50261184(5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to mouse gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483177(CHEMBL1632175)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483190(CHEMBL1632170)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50261184(5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to rat gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Drug Discovery Laboratory

Curated by ChEMBL
LigandPNGBDBM50483189(CHEMBL1632176)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]GR113808 from human 5HT4 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50261184(5-((3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaphth...)
Affinity DataKi:  6nMAssay Description:Binding affinity to human gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50224310(5-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human gonadotropin-releasing hormone receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Norwegian Medical Cyclotron Centre

Curated by ChEMBL
LigandPNGBDBM50009297(CHEMBL3233520)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]Triptorelin from rat full-length gonadotropin-releasing hormone receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
University Of Oslo

Curated by ChEMBL
LigandPNGBDBM50442804(CHEMBL2440452)
Affinity DataKi:  63nMAssay Description:Displacement of [125I]SB207710 from 5-HT4 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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