Affinity DataIC50: 2.80nMAssay Description:Inhibition of GST-tagged human full-length CHK1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant His6-tagged PIM1 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of ATP measured after 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of Pim-1 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human Pim3 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 12.4nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant His6-tagged PIM3 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant rat DYRK1A (1 to 499 residues ) expressed in bacterial expression system using KKISGRLSPIMTEQ as substrate measured after 3...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human plasmin using pyroGlu-Phe-Lys-pNA.HClMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of full-length human Pim-3 using RSRHSSYPAG as substrate incubated in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of full-length human PIM3 using RSRHSSYPAGT as substrate assessed as residual kinase activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of ATP measured after 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of BRD9 (unknown origin) incubated in dark for 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human full length (His)6-tagged Pim-3 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of BRD9 (unknown origin) incubated in dark for 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of human Chk1More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of Pim-3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of human Chk1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using myelin basic protein as substrate incubated for 30 mins in presen...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human PIM1 expressed in bacterial expression system using histone H1 as substrate measured after 30 mins in presence of ATP...More data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of full-length human Pim-1 using RSRHSSYPAG as substrate incubated in presence of [gamma33P]ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human full length Pim-3 using RSRHSSYPAGT as substrate assessed as residual activity after 30 mins in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant mouse CLK1 expressed in bacteria using GRSRSRSRSRSR as substrate in presence of ATP measured after 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human PIM1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition assay using PIM-1, PIM-2 and PIM-3.More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL