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Found 40 with Last Name = 'antal zimanyi' and Initial = 'i'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataIC50:  9nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136366((S)-Piperidine-3-carboxylic acid [(R)-1-(4-chloro-...)
Affinity DataIC50:  9nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136365(CHEMBL337571 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataIC50:  10nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136357(CHEMBL341982 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataIC50:  10nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136372(CHEMBL343076 | N-{2-[(R)-1-(4-Chloro-benzyl)-2-(4-...)
Affinity DataIC50:  11nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136367(CHEMBL137273 | N-{2-[(R)-1-(4-Chloro-benzyl)-2-(4-...)
Affinity DataIC50:  12nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136360(3-Acetylamino-N-[(R)-1-(4-chloro-benzyl)-2-(4-cycl...)
Affinity DataIC50:  12nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136364((R)-Piperidine-3-carboxylic acid [(R)-1-(4-chloro-...)
Affinity DataIC50:  12nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136370(3-Benzylamino-N-[(R)-1-(4-chloro-benzyl)-2-(4-cycl...)
Affinity DataIC50:  14nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136355(3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-(4-cyclohexyl...)
Affinity DataIC50:  16nMAssay Description:Stimulation of adenylate cyclase in HEK293 cells expressing the human MC4R receptor was determined by measuring cAMP accumulation using the RPA559 SP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136368(Azetidine-3-carboxylic acid [(R)-1-(4-chloro-benzy...)
Affinity DataIC50:  16nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136363(3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-(4-cyclohexyl...)
Affinity DataIC50:  18nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136356(CHEMBL343742 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataIC50:  21nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136369((S)-Piperidine-3-carboxylic acid {2-[(R)-1-(4-chlo...)
Affinity DataIC50:  22nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136371(CHEMBL343720 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataIC50:  22nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136361((R)-Piperidine-3-carboxylic acid {2-[(R)-1-(4-chlo...)
Affinity DataIC50:  25nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136362(3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-(4-cyclohexyl...)
Affinity DataIC50:  30nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136359(CHEMBL136366 | N-{2-[(R)-1-(4-Chloro-benzyl)-2-(4-...)
Affinity DataIC50:  90nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136373(CHEMBL340959 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataIC50:  110nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136358(CHEMBL137318 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataIC50:  180nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135642(Benzo[b]thiophene-2-carboxylic acid (2-benzylsulfa...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135647(CHEMBL328861 | N-(2-Benzylsulfanyl-phenyl)-N-(3-di...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135642(Benzo[b]thiophene-2-carboxylic acid (2-benzylsulfa...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135642(Benzo[b]thiophene-2-carboxylic acid (2-benzylsulfa...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135638(Benzo[b]thiophene-2-carboxylic acid (2-butyl-pheny...)
Affinity DataIC50:  2.20E+3nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135646((1R,2R)-2-Phenyl-cyclopropanecarboxylic acid (2-be...)
Affinity DataIC50:  3.70E+3nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135651(Benzo[b]thiophene-2-carboxylic acid biphenyl-2-yl-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135650(Benzo[b]thiophene-2-carboxylic acid (2-benzylsulfa...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135649(Benzo[b]thiophene-2-carboxylic acid (3-dimethylami...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135644(Benzo[b]thiophene-2-carboxylic acid (2-benzoylamin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135645((E)-N-(2-Benzylsulfanyl-phenyl)-N-(3-dimethylamino...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135643(Benzo[b]thiophene-2-carboxylic acid (2-benzylsulfa...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135641(Benzo[b]thiophene-2-carboxylic acid (2-benzyl-phen...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135640(3-Chloro-benzo[b]thiophene-2-carboxylic acid (2-be...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135639(Benzofuran-2-carboxylic acid (2-benzylsulfanyl-phe...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135648(Benzo[b]thiophene-2-carboxylic acid (2-benzylsulfa...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against SMS-KAN cell membranes endogenously expressing Neuropeptide Y receptor type 2 using [125I]-PYY as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136357(CHEMBL341982 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataEC50:  40nMAssay Description:Stimulation of adenylate cyclase in HEK293 cells expressing the human MC4R receptor was determined by measuring cAMP accumulation using the RPA559 SP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136365(CHEMBL337571 | N-[(R)-1-(4-Chloro-benzyl)-2-(4-cyc...)
Affinity DataEC50:  70nMAssay Description:Binding activity was measured using membranes of Hi5 cells expressing the human MC4R receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50136355(3-Amino-N-[(R)-1-(4-chloro-benzyl)-2-(4-cyclohexyl...)
Affinity DataEC50:  170nMAssay Description:Stimulation of adenylate cyclase in HEK293 cells expressing the human MC4R receptor was determined by measuring cAMP accumulation using the RPA559 SP...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataEC50:  3.60nMAssay Description:Stimulation of adenylate cyclase in HEK293 cells expressing the human MC4R receptor was determined by measuring cAMP accumulation using the RPA559 SP...More data for this Ligand-Target Pair