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Found 15 with Last Name = 'antemano' and Initial = 'r'
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335603(CHEMBL1651095 | Pulicatin A)
Affinity DataKi:  505nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335599(CHEMBL1651091 | pulicatins F)
Affinity DataKi:  1.03E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335600(CHEMBL1651092 | pulicatins G)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335598(CHEMBL1651090 | aerugine)
Affinity DataKi:  1.36E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335604(CHEMBL1651096 | pulicatin D)
Affinity DataKi:  1.54E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335601(CHEMBL1651093 | Watasemycins A)
Affinity DataKi:  3.92E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335602(CHEMBL1651094 | Watasemycins B)
Affinity DataKi:  4.70E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345471((R)-N-((S)-1-((6S,9S,12R,13R,Z)-3-ethylidene-9-iso...)
Affinity DataIC50:  2.27E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345471((R)-N-((S)-1-((6S,9S,12R,13R,Z)-3-ethylidene-9-iso...)
Affinity DataIC50:  2.27E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345472(CHEMBL1784750 | Nobilamide B)
Affinity DataIC50:  2.75E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345472(CHEMBL1784750 | Nobilamide B)
Affinity DataIC50:  2.75E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345473((R)-2-((R)-2-acetamido-3-phenylpropanamido)-N-((S)...)
Affinity DataIC50:  1.32E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345473((R)-2-((R)-2-acetamido-3-phenylpropanamido)-N-((S)...)
Affinity DataIC50:  1.32E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345474(CHEMBL1784749 | Nobilamide A)
Affinity DataIC50:  1.67E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50345474(CHEMBL1784749 | Nobilamide A)
Affinity DataIC50:  1.67E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed