Affinity DataKi: 505nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.03E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.54E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.92E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.27E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.27E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.75E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.75E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.32E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.32E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.67E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.67E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair