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Found 51 with Last Name = 'antunes' and Initial = 'oa'
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataKi:  1.80E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataKi:  3.00E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataKi:  7.04E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataKi:  7.07E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataKi:  7.19E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataKi:  7.51E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataKi:  7.74E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataKi:  8.03E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataKi:  2.00E+5nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataKi:  3.57E+5nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481018(CHEMBL568883)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481028(CHEMBL566620)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481036(CHEMBL568589)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481029(CHEMBL569671)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481014(CHEMBL568951)
Affinity DataIC50:  0.339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481020(CHEMBL565964)
Affinity DataIC50:  0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481023(CHEMBL566849)
Affinity DataIC50:  0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481040(CHEMBL566842)
Affinity DataIC50:  0.501nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481024(CHEMBL566902)
Affinity DataIC50:  0.741nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481017(CHEMBL568840)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481015(CHEMBL568832)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481025(CHEMBL567444)
Affinity DataIC50:  0.851nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481033(CHEMBL565528)
Affinity DataIC50:  0.891nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481035(CHEMBL569670)
Affinity DataIC50:  1nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481037(CHEMBL569236)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481032(CHEMBL569569)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481022(CHEMBL568365)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM586099(BDBM50064200 | TL-3)
Affinity DataIC50:  2nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481019(CHEMBL571731)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481031(CHEMBL567043)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481041(CHEMBL569673)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481016(CHEMBL568817)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481038(CHEMBL568977)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM198((2S)-N-[(2S,3S,4S,5S)-3,4-dihydroxy-5-[(2S)-3-meth...)
Affinity DataIC50:  15nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481027(CHEMBL566839)
Affinity DataIC50:  18nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481030(CHEMBL570827)
Affinity DataIC50:  22nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481013(CHEMBL569111)
Affinity DataIC50:  38nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481034(CHEMBL567500)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481021(CHEMBL565766)
Affinity DataIC50:  141nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481039(CHEMBL569672)
Affinity DataIC50:  339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481026(CHEMBL569573)
Affinity DataIC50:  363nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataIC50:  1.63E+4nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391078(CHEMBL2087346)
Affinity DataIC50:  9.91E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391075(CHEMBL2087343)
Affinity DataIC50:  9.92E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391079(CHEMBL2087347)
Affinity DataIC50:  1.61E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataIC50:  1.96E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-7(Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391076(CHEMBL2087344)
Affinity DataIC50:  2.05E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro

Curated by ChEMBL
LigandPNGBDBM50391077(CHEMBL2087345)
Affinity DataIC50:  3.24E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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