Affinity DataKi: 1.80E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 7.04E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 7.07E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 7.19E+4nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.51E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.74E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8.03E+4nMAssay Description:Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 2.00E+5nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataKi: 3.57E+5nMAssay Description:Competitive inhibition of human KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.501nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.741nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.851nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 0.891nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 141nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras
Curated by ChEMBL
Universidade Federal De Lavras
Curated by ChEMBL
Affinity DataIC50: 363nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataIC50: 9.91E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataIC50: 9.92E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.61E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.96E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.05E+5nMAssay Description:Inhibition of human recombinant KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Universidade Federal Do Tri£Ngulo Mineiro
Curated by ChEMBL
Affinity DataIC50: 3.24E+5nMAssay Description:Inhibition of human recombinant KLK5 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by FRET analysisMore data for this Ligand-Target Pair