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Found 100 with Last Name = 'anzai' and Initial = 'm'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataIC50: <1nMAssay Description:Inhibition of recombinant wild type EGFR (696 to C terminal end) (unknown origin) using poly (Glu-Tyr) as substrate preincubated for 30 mins followed...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50559514(CHEMBL4791596)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of recombinant wild type EGFR T790M/L858R mutant (696 to C terminal end) (unknown origin) using poly (Glu-Tyr) as substrate preincubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of recombinant wild type EGFR T790M/L858R mutant (696 to C terminal end) (unknown origin) using poly (Glu-Tyr) as substrate preincubated f...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant wild type EGFR (696 to C terminal end) (unknown origin) using poly (Glu-Tyr) as substrate preincubated for 30 mins followed...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50559514(CHEMBL4791596)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of recombinant wild type EGFR (696 to C terminal end) (unknown origin) using poly (Glu-Tyr) as substrate preincubated for 30 mins followed...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nagasaki University

Curated by ChEMBL
LigandPNGBDBM50559511(CHEMBL4746895)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of recombinant wild type EGFR T790M/L858R mutant (696 to C terminal end) (unknown origin) using poly (Glu-Tyr) as substrate preincubated f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411106(CHEMBL387098)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411105(CHEMBL216037)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411176(CHEMBL383850)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411164(CHEMBL386412)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411143(CHEMBL384614)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411137(CHEMBL383910)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411132(CHEMBL213868)
Affinity DataIC50:  6nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411150(CHEMBL387220)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411115(CHEMBL217924)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411161(CHEMBL385205)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411133(CHEMBL385705)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411124(CHEMBL217385)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411159(CHEMBL214978)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411158(CHEMBL385707)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411157(CHEMBL215164)
Affinity DataIC50:  6.20nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411120(CHEMBL218565)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411126(CHEMBL384370)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411127(CHEMBL214500)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411165(CHEMBL215360)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411110(CHEMBL215306)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411184(CHEMBL215239)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411169(CHEMBL383902)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411183(CHEMBL217447)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411111(CHEMBL385342)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411174(CHEMBL384929)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411136(CHEMBL385926)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411182(CHEMBL387281)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411142(CHEMBL217417)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411104(CHEMBL217335)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411173(CHEMBL215968)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411167(CHEMBL215173)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411163(CHEMBL217030)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411154(CHEMBL214469)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411149(CHEMBL215518)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411135(CHEMBL386623)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411102(CHEMBL384538)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411128(CHEMBL215806)
Affinity DataIC50:  6.80nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411144(CHEMBL384020)
Affinity DataIC50:  6.80nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411178(CHEMBL410320)
Affinity DataIC50:  7.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411180(CHEMBL214662)
Affinity DataIC50:  7.70nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411114(CHEMBL213915)
Affinity DataIC50:  8.10nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411172(CHEMBL214135)
Affinity DataIC50:  8.10nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411151(CHEMBL217265)
Affinity DataIC50:  8.20nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Teikyo University

Curated by ChEMBL
LigandPNGBDBM50411168(CHEMBL387286)
Affinity DataIC50:  8.20nMAssay Description:Antagonist activity against 1-alpha,25-dihydroxy vitamin D3-induced HL60 cell differentiation by NBT reduction methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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