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Found 65 with Last Name = 'apelt' and Initial = 'j'
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110291((7-Chloro-quinolin-4-yl)-[4-(3-piperidin-1-yl-prop...)
Affinity DataKi:  0.0860nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110288(CHEMBL15153 | N-(4-(3-(piperidin-1-yl)propoxy)phen...)
Affinity DataKi:  0.0910nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110300(CHEMBL15056 | N-(4-(3-(piperidin-1-yl)propoxy)phen...)
Affinity DataKi:  0.330nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110311(CHEMBL276938 | {2-[4-(3-Piperidin-1-yl-propoxy)-ph...)
Affinity DataKi:  0.530nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110285(CHEMBL274041 | {3-[4-(3-Piperidin-1-yl-propoxy)-ph...)
Affinity DataKi:  0.75nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110299(CHEMBL14754 | {3-[4-(3-Piperidin-1-yl-propoxy)-phe...)
Affinity DataKi:  1.40nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110290(CHEMBL14484 | {4-[4-(3-Piperidin-1-yl-propoxy)-phe...)
Affinity DataKi:  1.5nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110306((6-Piperidin-1-yl-hexyl)-(1,2,3,4-tetrahydro-acrid...)
Affinity DataKi:  1.80nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110310((3-Methyl-quinolin-4-yl)-(6-piperidin-1-yl-hexyl)-...)
Affinity DataKi:  3.60nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110297((6-Piperidin-1-yl-hexyl)-quinolin-4-yl-amine; Oxal...)
Affinity DataKi:  7.60nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110312((7-Chloro-quinolin-4-yl)-(8-piperidin-1-yl-octyl)-...)
Affinity DataKi:  7.80nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110282((7-Chloro-quinolin-4-yl)-(7-piperidin-1-yl-heptyl)...)
Affinity DataKi:  9.90nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110289((7-Chloro-quinolin-4-yl)-(10-piperidin-1-yl-decyl)...)
Affinity DataKi:  12nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110294((5-Piperidin-1-yl-pentyl)-quinolin-4-yl-amine; Oxa...)
Affinity DataKi:  15nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110295((7-Chloro-quinolin-4-yl)-(6-piperidin-1-yl-hexyl)-...)
Affinity DataKi:  18nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110303((2-Piperidin-1-yl-ethyl)-(1,2,3,4-tetrahydro-acrid...)
Affinity DataKi:  19nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110304((7-Chloro-quinolin-4-yl)-(5-piperidin-1-yl-pentyl)...)
Affinity DataKi:  26nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110301((7-Chloro-quinolin-4-yl)-(12-piperidin-1-yl-dodecy...)
Affinity DataKi:  32nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110286((3-Piperidin-1-yl-propyl)-(1,2,3,4-tetrahydro-acri...)
Affinity DataKi:  34nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110281(CHEMBL14656 | Methyl-(3-piperidin-1-yl-propyl)-(1,...)
Affinity DataKi:  50nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110307((3-Methyl-quinolin-4-yl)-(3-piperidin-1-yl-propyl)...)
Affinity DataKi:  70nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110292(CHEMBL14781 | Methyl-(2-piperidin-1-yl-ethyl)-(1,2...)
Affinity DataKi:  78nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110283((7-Chloro-quinolin-4-yl)-(4-piperidin-1-yl-butyl)-...)
Affinity DataKi:  82nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110287((3-Piperidin-1-yl-propyl)-quinolin-4-yl-amine; Oxa...)
Affinity DataKi:  85nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110284((4-Piperidin-1-yl-butyl)-quinolin-4-yl-amine; Oxal...)
Affinity DataKi:  90nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110302(Acridin-9-yl-(3-piperidin-1-yl-propyl)-amine; Oxal...)
Affinity DataKi:  188nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110313((2-Piperidin-1-yl-ethyl)-quinolin-4-yl-amine; Oxal...)
Affinity DataKi:  191nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110293(CHEMBL14860 | Methyl-(2-piperidin-1-yl-ethyl)-quin...)
Affinity DataKi:  362nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110305((7-Chloro-quinolin-4-yl)-(3-piperidin-1-yl-propyl)...)
Affinity DataKi:  378nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110309(CHEMBL14740 | Methyl-(3-piperidin-1-yl-propyl)-qui...)
Affinity DataKi:  411nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110298(CHEMBL277113 | Ethyl-(3-piperidin-1-yl-propyl)-qui...)
Affinity DataKi:  1.13E+3nMAssay Description:Affinity for displacement of [125I]-iodoproxyfan from human histamine H3 receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110309(CHEMBL14740 | Methyl-(3-piperidin-1-yl-propyl)-qui...)
Affinity DataIC50:  16nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110306((6-Piperidin-1-yl-hexyl)-(1,2,3,4-tetrahydro-acrid...)
Affinity DataIC50:  21nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110285(CHEMBL274041 | {3-[4-(3-Piperidin-1-yl-propoxy)-ph...)
Affinity DataIC50:  31nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110303((2-Piperidin-1-yl-ethyl)-(1,2,3,4-tetrahydro-acrid...)
Affinity DataIC50:  34nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110286((3-Piperidin-1-yl-propyl)-(1,2,3,4-tetrahydro-acri...)
Affinity DataIC50:  45nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110296(CHEMBL14868 | {4-[4-(3-Piperidin-1-yl-propoxy)-phe...)
Affinity DataIC50:  48nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110300(CHEMBL15056 | N-(4-(3-(piperidin-1-yl)propoxy)phen...)
Affinity DataIC50:  48nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110298(CHEMBL277113 | Ethyl-(3-piperidin-1-yl-propyl)-qui...)
Affinity DataIC50:  49nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110288(CHEMBL15153 | N-(4-(3-(piperidin-1-yl)propoxy)phen...)
Affinity DataIC50:  51nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110294((5-Piperidin-1-yl-pentyl)-quinolin-4-yl-amine; Oxa...)
Affinity DataIC50:  53nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110284((4-Piperidin-1-yl-butyl)-quinolin-4-yl-amine; Oxal...)
Affinity DataIC50:  64nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110287((3-Piperidin-1-yl-propyl)-quinolin-4-yl-amine; Oxa...)
Affinity DataIC50:  64nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110290(CHEMBL14484 | {4-[4-(3-Piperidin-1-yl-propoxy)-phe...)
Affinity DataIC50:  73nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110297((6-Piperidin-1-yl-hexyl)-quinolin-4-yl-amine; Oxal...)
Affinity DataIC50:  84nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110299(CHEMBL14754 | {3-[4-(3-Piperidin-1-yl-propoxy)-phe...)
Affinity DataIC50:  95nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110302(Acridin-9-yl-(3-piperidin-1-yl-propyl)-amine; Oxal...)
Affinity DataIC50:  110nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  110nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110282((7-Chloro-quinolin-4-yl)-(7-piperidin-1-yl-heptyl)...)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Rattus norvegicus)
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50110293(CHEMBL14860 | Methyl-(2-piperidin-1-yl-ethyl)-quin...)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat kidney Histamine N-Methyltransferase (HMT) activity determined by the formation of N-methylhistamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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