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Found 67 with Last Name = 'appella' and Initial = 'dh'
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481913(CHEMBL1075826)
Affinity DataIC50:  900nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35079(N-acylpolyamine (NAPA) scaffold, 26)
Affinity DataIC50:  2.30E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35078(N-acylpolyamine (NAPA) scaffold, 25)
Affinity DataIC50:  2.60E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35078(N-acylpolyamine (NAPA) scaffold, 25)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35076(N-acylpolyamine (NAPA) scaffold, 23)
Affinity DataIC50:  2.80E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35077(N-acylpolyamine (NAPA) scaffold, 24)
Affinity DataIC50:  2.80E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35080(N-acylpolyamine (NAPA) scaffold, 27)
Affinity DataIC50:  2.90E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35079(N-acylpolyamine (NAPA) scaffold, 26)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35076(N-acylpolyamine (NAPA) scaffold, 23)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35080(N-acylpolyamine (NAPA) scaffold, 27)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35083(N-acylpolyamine (NAPA) scaffold, 34)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481920(CHEMBL1075815)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35071(N-acylpolyamine (NAPA) scaffold, 18)
Affinity DataIC50:  6.40E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35071(N-acylpolyamine (NAPA) scaffold, 18)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35074(N-acylpolyamine (NAPA) scaffold, 21)
Affinity DataIC50:  6.60E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481917(CHEMBL1075830)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35077(N-acylpolyamine (NAPA) scaffold, 24)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35070(N-acylpolyamine (NAPA) scaffold, 17)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35072(N-acylpolyamine (NAPA) scaffold, 19)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35074(N-acylpolyamine (NAPA) scaffold, 21)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35069(N-acylpolyamine (NAPA) scaffold, 16)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35070(N-acylpolyamine (NAPA) scaffold, 17)
Affinity DataIC50:  8.20E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35075(N-acylpolyamine (NAPA) scaffold, 22)
Affinity DataIC50:  8.20E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35062(N-acylpolyamine (NAPA) scaffold, 9)
Affinity DataIC50:  9.20E+3nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35073(N-acylpolyamine (NAPA) scaffold, 20)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35075(N-acylpolyamine (NAPA) scaffold, 22)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35069(N-acylpolyamine (NAPA) scaffold, 16)
Affinity DataIC50:  1.00E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481915(CHEMBL1075824)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35072(N-acylpolyamine (NAPA) scaffold, 19)
Affinity DataIC50:  1.05E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35068(N-acylpolyamine (NAPA) scaffold, 15)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35068(N-acylpolyamine (NAPA) scaffold, 15)
Affinity DataIC50:  1.20E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481919(CHEMBL1075821)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35081(N-acylpolyamine (NAPA) scaffold, 28)
Affinity DataIC50:  1.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35066(N-acylpolyamine (NAPA) scaffold, 13)
Affinity DataIC50:  1.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35066(N-acylpolyamine (NAPA) scaffold, 13)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35067(N-acylpolyamine (NAPA) scaffold, 14)
Affinity DataIC50:  1.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35081(N-acylpolyamine (NAPA) scaffold, 28)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481914(CHEMBL1075825)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35061(N-acylpolyamine (NAPA) scaffold, 8)
Affinity DataIC50:  1.70E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35073(N-acylpolyamine (NAPA) scaffold, 20)
Affinity DataIC50:  1.70E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35058(N-acylpolyamine (NAPA) scaffold, 5)
Affinity DataIC50:  1.80E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481918(CHEMBL1081563)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35067(N-acylpolyamine (NAPA) scaffold, 14)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35059(N-acylpolyamine (NAPA) scaffold, 6)
Affinity DataIC50:  2.00E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35063(N-acylpolyamine (NAPA) scaffold, 10)
Affinity DataIC50:  2.40E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35062(N-acylpolyamine (NAPA) scaffold, 9)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481921(CHEMBL1075829)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481916(CHEMBL1075823)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Nih

LigandPNGBDBM35063(N-acylpolyamine (NAPA) scaffold, 10)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Nih

LigandPNGBDBM35060(N-acylpolyamine (NAPA) scaffold, 7)
Affinity DataIC50:  3.80E+4nMpH: 7.6 T: 2°CAssay Description:Inhibitory activities of NAPAs were measured by fluorescence anisotropy competition experiments. Protein was incubated with fluorescein-labeled huma...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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