TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 170nM ΔG°: -38.2kJ/mole IC50: 390nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetSerine/threonine-protein kinase Sgk1(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 400nM ΔG°: -36.2kJ/mole IC50: 500nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 740nM ΔG°: -34.6kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 1.18E+3nM ΔG°: -33.5kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 1.85E+3nM ΔG°: -32.4kJ/mole IC50: 890nMpH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
Affinity DataKi: 4.50E+3nM ΔG°: -30.2kJ/molepH: 7.5 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of 100 uM ATP/ [gam...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
University Of Dundee
Curated by PDSP Ki Database
University Of Dundee
Curated by PDSP Ki Database
Target3-phosphoinositide-dependent protein kinase 1 [51-359](Homo sapiens (Human))
University Of Dundee
University Of Dundee
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:In vitro PDK1 assay using purified enzyme, was incubated with substrate PDKtide, and test compounds in the presence of ATP/ [gamma-32P] ATP. 32P inco...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-359](Homo sapiens (Human))
University Of Dundee
University Of Dundee
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:In vitro PDK1 assay using purified enzyme, was incubated with substrate PDKtide, and test compounds in the presence of ATP/ [gamma-32P] ATP. 32P inco...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-359](Homo sapiens (Human))
University Of Dundee
University Of Dundee
Affinity DataIC50: 6.5nMpH: 7.5 T: 2°CAssay Description:In vitro PDK1 assay using purified enzyme, was incubated with substrate PDKtide, and test compounds in the presence of ATP/ [gamma-32P] ATP. 32P inco...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by ChEMBL
University Of Dundee
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of CAMKKbeta in the presence of 20uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 12.4nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] labe...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Aurora C in the presence of 5uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMpH: 7.5 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] labe...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by ChEMBL
University Of Dundee
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of RIP2 in the presence of 100uM ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of Aurora B in the presence of 20uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMpH: 7.5 T: 2°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-33P] labe...More data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by ChEMBL
University Of Dundee
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of RIP2 in the presence of 100uM ATPMore data for this Ligand-Target Pair
TargetReceptor-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by ChEMBL
University Of Dundee
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of RIP2 in the presence of 100uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University Of Dundee
Curated by ChEMBL
University Of Dundee
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK2-cyclinA in the presence of 20uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université
Curated by ChEMBL
Clermont Université
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of PIM3 in the presence of 5uM ATPMore data for this Ligand-Target Pair