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Found 1085 with Last Name = 'barth' and Initial = 'm'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420581(CHEMBL2087422)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50326708(CHEMBL1254771 | N-(4-(4,5-dihydro-1H-imidazol-2-yl...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420570(CHEMBL2087434)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420569(CHEMBL2087433)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420579(CHEMBL2087423)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420589(CHEMBL2087031)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420580(CHEMBL2087421)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420603(CHEMBL2087035)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420595(CHEMBL2087409)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420597(CHEMBL2087411)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420582(CHEMBL2087420)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420573(CHEMBL2087429)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420571(CHEMBL2087432)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420601(CHEMBL2087412)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420598(CHEMBL2087413)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420577(CHEMBL2087424)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of M£Nster

Curated by ChEMBL
LigandPNGBDBM50112086(3-({2-[(4-Carbamimidoyl-phenylamino)-methyl]-1-met...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of human coagulation factor alpha-thrombin using Boc-Val-Pro-Arg-AMC as fluorogenic substrate measured at 1 min interval for 1 hr by fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420568(CHEMBL2087435)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420596(CHEMBL2087410)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420583(CHEMBL2087418)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420574(CHEMBL2087427)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420600(CHEMBL2087415)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420572(CHEMBL2087431)
Affinity DataKi:  9.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420575(CHEMBL2087428)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420576(CHEMBL2087426)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420594(CHEMBL2087036)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420593(CHEMBL2087034)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420586(CHEMBL2087430)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420584(CHEMBL2087419)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420591(CHEMBL2087029)
Affinity DataKi:  59nMAssay Description:Binding affinity to B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420599(CHEMBL2087414)
Affinity DataKi:  63.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420592(CHEMBL2087033)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420567(CHEMBL2087436)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420585(CHEMBL2087417)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420590(CHEMBL2087030)
Affinity DataKi:  100nMAssay Description:Binding affinity to B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420578(CHEMBL2087425)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420588(CHEMBL2087027)
Affinity DataKi:  130nMAssay Description:Binding affinity to B2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420602(CHEMBL2087416)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051375((6S,8aS)-5,5,8a-Trimethyl-2-((E)-1,5,9-trimethyl-d...)
Affinity DataKi:  300nMAssay Description:Binding affinity towards competitive inhibition against rat microsomal Oxidosqualene-lanosterol cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50051375((6S,8aS)-5,5,8a-Trimethyl-2-((E)-1,5,9-trimethyl-d...)
Affinity DataKi:  400nMAssay Description:Binding affinity towards noncompetetive inhibition against rat microsomal Oxidosqualene-lanosterol cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420587(CHEMBL2087028)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity to B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420588(CHEMBL2087027)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity to B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of M£Nster

Curated by ChEMBL
LigandPNGBDBM50112086(3-({2-[(4-Carbamimidoyl-phenylamino)-methyl]-1-met...)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of human coagulation factor Xa using Boc-Ile-Glu-Gly-Arg-AMC as fluorogenic substrate measured at 1 min interval for 1 hr by fluorometric ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Laboratoires Fournier

Curated by ChEMBL
LigandPNGBDBM50420587(CHEMBL2087028)
Affinity DataKi:  4.30E+4nMAssay Description:Binding affinity to B2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50544830(CHEMBL4635876)
Affinity DataIC50: >0.158nMAssay Description:Inhibition of JAK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50585527(CHEMBL5084861)
Affinity DataIC50: >0.158nMAssay Description:Inhibition of GST-tagged recombinant human JAK2 (808 to 1132 residues) expressed in baculovirus expression system using ULight-JAK-1 Tyr1023 peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50585514(CHEMBL5086526)
Affinity DataIC50:  0.158nMAssay Description:Inhibition of GST-fused human JAK3 (810 to 1100 residues) expressed in insect cells using ULight-JAK-1 Tyr1023 peptide as substrate preincubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50585515(CHEMBL5076189)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of GST-fused human JAK3 (810 to 1100 residues) expressed in insect cells using ULight-JAK-1 Tyr1023 peptide as substrate preincubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50544831(CHEMBL4634979)
Affinity DataIC50:  0.251nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50544830(CHEMBL4635876)
Affinity DataIC50:  0.316nMAssay Description:Inhibition of JAK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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