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Found 47 with Last Name = 'bhatnagar' and Initial = 'rk'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.0450nMAssay Description:Binding affinity of compound against Dopamine receptor D2 binding site using radioligand [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity of compound against 5-hydroxytryptamine 1A receptor binding site using radioligand [3H]8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50017514(8,11-Dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dib...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity of compound against 5-hydroxytryptamine 1A receptor binding site using radioligand [3H]8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  30nMAssay Description:Binding affinity of compound against 5-hydroxytryptamine 1A receptor binding site using radioligand [3H]8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50017514(8,11-Dimethoxy-6-methyl-5,6,6a,7-tetrahydro-4H-dib...)
Affinity DataKi:  210nMAssay Description:Binding affinity of compound against Dopamine receptor D2 binding site using radioligand [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50017513(8,11-Dimethoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dib...)
Affinity DataKi:  240nMAssay Description:Binding affinity of compound against 5-hydroxytryptamine 1A receptor binding site using radioligand [3H]8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50017513(8,11-Dimethoxy-6-propyl-5,6,6a,7-tetrahydro-4H-dib...)
Affinity DataKi:  770nMAssay Description:Binding affinity of compound against Dopamine receptor D2 binding site using radioligand [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
College Of Pharmacy University Of Iowa

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding affinity of compound against Dopamine receptor D2 binding site using radioligand [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFalcipain 2(Plasmodium falciparum)
International Center For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50261135(CHEMBL525938 | LMNNAEHINQFYMFI)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant falcipain-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50368271(CHEMBL1204112)
Affinity DataIC50:  3nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50004000((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...)
Affinity DataIC50:  30nMAssay Description:Concentration required to inhibit hydrolytic activity of Acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50313079(3-Dimethylcarbamoyloxy-1-methyl-pyridinium; bromid...)
Affinity DataIC50:  50nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataIC50:  510nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataIC50:  830nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50224035(79907 | Lergotrile)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223956(CHEMBL555412)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50368269(CHEMBL1202156)
Affinity DataIC50:  6.90E+3nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50001955((-)6-Methyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]qu...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50368268(CHEMBL1202155)
Affinity DataIC50:  9.90E+3nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223901(CHEMBL544695)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223957(CHEMBL544931)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50107876((5,6-Dimethoxy-indan-2-yl)-dipropyl-amine | CHEMBL...)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50368272(CHEMBL1202157)
Affinity DataIC50:  1.42E+4nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290378(2-Dipropylamino-indan-5,6-diol | CHEMBL277743)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50012004((2-Biphenyl-4-yl-2-oxo-ethyl)-[1,3]dioxan-2-ylmeth...)
Affinity DataIC50:  2.01E+4nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50224035(79907 | Lergotrile)
Affinity DataIC50:  2.37E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50368270(CHEMBL1202154)
Affinity DataIC50:  2.50E+4nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223959(CHEMBL538227)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50224033(CHEMBL540009)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50224034(CHEMBL538726)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223957(CHEMBL544931)
Affinity DataIC50:  5.39E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223901(CHEMBL544695)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50011998(CHEMBL298102 | [1,3]Dioxan-2-ylmethyl-dimethyl-(2-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50011996(CHEMBL290329 | [1,3]Dioxan-2-ylmethyl-trimethyl-am...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit hydrolytic activity of bovine erythrocyte acetylcholinesterase by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223900(CHEMBL34176)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223956(CHEMBL555412)
Affinity DataIC50:  1.04E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223958(CHEMBL544697)
Affinity DataIC50:  1.05E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50224033(CHEMBL540009)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50224036(CHEMBL543991)
Affinity DataIC50:  2.46E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]spiperone as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50224034(CHEMBL538726)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290378(2-Dipropylamino-indan-5,6-diol | CHEMBL277743)
Affinity DataIC50:  4.12E+5nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223959(CHEMBL538227)
Affinity DataIC50:  1.66E+6nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223900(CHEMBL34176)
Affinity DataIC50:  2.30E+6nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50223958(CHEMBL544697)
Affinity DataIC50:  5.10E+7nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50107876((5,6-Dimethoxy-indan-2-yl)-dipropyl-amine | CHEMBL...)
Affinity DataIC50:  1.47E+8nMAssay Description:Inhibitory binding activity against dopamine receptor using [3H]ADTN as the radioligand in striatal tissue of calf brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeme ligase(Plasmodium falciparum (isolate 3D7))
International Centre For Genetic Engineering And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50250134(CHEMBL4068384)
Affinity DataKd:  2.96E+3nMAssay Description:Binding affinity to Plasmodium falciparum 3D7 HDP assessed as equilibrium dissociation constant by SPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed