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Found 482 with Last Name = 'bobko' and Initial = 'ma'
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030096((R)-11-{Hydroxy-[4-methoxy-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030095((R)-11-{Hydroxy-[4-methoxy-3-(2-methyl-butyl)-phen...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030095((R)-11-{Hydroxy-[4-methoxy-3-(2-methyl-butyl)-phen...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030096((R)-11-{Hydroxy-[4-methoxy-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030099((R)-5-(1H-Indol-3-ylmethyl)-17-isopropyl-11-[4-met...)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030092((R)-11-{Hydroxy-[4-hydroxy-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030092((R)-11-{Hydroxy-[4-hydroxy-3-(3-methyl-but-2-enyl)...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030094((R)-11-[Hydroxy-(4-methoxy-phenyl)-methyl]-5-(1H-i...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030094((R)-11-[Hydroxy-(4-methoxy-phenyl)-methyl]-5-(1H-i...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50407271(CHEMBL2112592)
Affinity DataKi:  2.70E+4nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50407272(CHEMBL2111789)
Affinity DataKi:  3.10E+4nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50407271(CHEMBL2112592)
Affinity DataKi:  4.80E+4nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030091((R)-5-(1H-Indol-3-ylmethyl)-17-isopropyl-11-(4-met...)
Affinity DataKi:  7.20E+4nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030091((R)-5-(1H-Indol-3-ylmethyl)-17-isopropyl-11-(4-met...)
Affinity DataKi:  7.30E+4nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50407272(CHEMBL2111789)
Affinity DataKi:  9.30E+4nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030097((R)-11-[Hydroxy-(4-hydroxy-phenyl)-methyl]-5-(1H-i...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030097((R)-11-[Hydroxy-(4-hydroxy-phenyl)-methyl]-5-(1H-i...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030098((R)-11-(4-Hydroxy-benzyl)-5-(1H-indol-3-ylmethyl)-...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030090((R)-11-(1H-Indol-5-ylmethyl)-5-(1H-indol-3-ylmethy...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030090((R)-11-(1H-Indol-5-ylmethyl)-5-(1H-indol-3-ylmethy...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]-NKA substance P binding to human urinary bladder membrane protein (NK2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50030098((R)-11-(4-Hydroxy-benzyl)-5-(1H-indol-3-ylmethyl)-...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [125I]- substance P binding to human astrocytoma cells (NK1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383996(CHEMBL2032134)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383999(CHEMBL2032137)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383966(CHEMBL2032148)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383998(CHEMBL2032136)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50384000(CHEMBL2032138)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383997(CHEMBL2032135)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383994(CHEMBL2032132)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383987(CHEMBL2032125)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383982(CHEMBL2032119)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383995(CHEMBL2032133)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383988(CHEMBL2032126)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383993(CHEMBL2032131)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50384003(CHEMBL2032142)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383968(CHEMBL2032140)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50384002(CHEMBL2032141)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383972(CHEMBL2032146)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383969(CHEMBL2032143)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383980(CHEMBL2032117)
Affinity DataIC50:  0.430nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383992(CHEMBL2032130)
Affinity DataIC50:  0.440nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383965(CHEMBL2032129)
Affinity DataIC50:  0.460nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383967(CHEMBL2032122)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383981(CHEMBL2032118)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383986(CHEMBL2032124)
Affinity DataIC50:  0.510nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383985(CHEMBL2032123)
Affinity DataIC50:  0.520nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383996(CHEMBL2032134)
Affinity DataIC50:  0.520nMAssay Description:Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383984(CHEMBL2032121)
Affinity DataIC50:  0.540nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50341250(CHEMBL1765751 | N-{(3R,5R)-1-[2-Amino-6-(3-amino-1...)
Affinity DataIC50:  0.631nMAssay Description:Inhibition of PDK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383989(CHEMBL2032127)
Affinity DataIC50:  0.660nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383978(CHEMBL2032115)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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