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Found 28 with Last Name = 'boyd' and Initial = 'rj'
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045092(5-(2-Carboxy-ethyl)-6-[(E)-6-(4-methoxy-phenyl)-he...)
Affinity DataKi:  5.90nMAssay Description:Inhibition constant against binding of [3H]-LTB4 to human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001611((E)-3-{3-(2-Carboxy-ethyl)-4-[6-(4-methoxy-phenyl)...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of binding of [3H]-LTB4 to receptor on nonradioactive LTB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039472(7-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-phenox...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039467(3-(3-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-phe...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045092(5-(2-Carboxy-ethyl)-6-[(E)-6-(4-methoxy-phenyl)-he...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of specific binding of LTB4 ( 0.1 nM) to receptors on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50029490(4-Ethyl-5-[6-methyl-6-(1H-tetrazol-5-yl)-heptyloxy...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039478(4-Ethyl-2-(1-methyl-1H-pyrazol-3-yl)-5-[6-methyl-6...)
Affinity DataIC50:  9.30nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039471((3-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-pheno...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039480((2-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-pheno...)
Affinity DataIC50:  12nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001611((E)-3-{3-(2-Carboxy-ethyl)-4-[6-(4-methoxy-phenyl)...)
Affinity DataIC50:  13nMAssay Description:Inhibition of specific binding of [3H]-LTB4 ( 0.1 nM) to LTB4 receptor on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039475(3-(4-{5-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-phe...)
Affinity DataIC50:  28nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045091(5-(2-Carboxy-ethyl)-6-decyloxy-9-oxo-9H-xanthene-2...)
Affinity DataIC50:  43nMAssay Description:Inhibition of specific binding of LTB4 ( 0.1 nM) to receptors on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039477((4-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-pheno...)
Affinity DataIC50:  54nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039469((4-{5-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-pheno...)
Affinity DataIC50:  55nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039470(4-{5-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-phenox...)
Affinity DataIC50:  82nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM81519(CAS_117690-79-6 | CGS 23356 | CHEMBL15766 | LY 255...)
Affinity DataIC50:  85.1nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039468(3-(4-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-phe...)
Affinity DataIC50:  87nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039476(4-Ethyl-2-(2-methyl-2H-pyrazol-3-yl)-5-[6-methyl-6...)
Affinity DataIC50:  107nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045092(5-(2-Carboxy-ethyl)-6-[(E)-6-(4-methoxy-phenyl)-he...)
Affinity DataIC50:  133nMAssay Description:The antagonist activity measured as inhibition of LTB4 response in aggregation of neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045096(3-[3-(2-Carboxy-ethyl)-4-decyloxy-benzoyl]-benzoic...)
Affinity DataIC50:  210nMAssay Description:Inhibition of specific binding of LTB4 ( 0.1 nM) to receptors on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039473(7-{3-[4-((E)-3-Dimethylamino-acryloyl)-2-ethyl-5-h...)
Affinity DataIC50:  319nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045091(5-(2-Carboxy-ethyl)-6-decyloxy-9-oxo-9H-xanthene-2...)
Affinity DataIC50:  513nMAssay Description:The antagonist activity measured as inhibition of LTB4 response in aggregation of neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039479(3-(3-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-phe...)
Affinity DataIC50:  738nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045093(7-(2-Carboxy-ethyl)-6-decyloxy-9-oxo-9H-xanthene-2...)
Affinity DataIC50:  832nMAssay Description:Inhibition of specific binding of LTB4 ( 0.1 nM) to receptors on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039481(3-(3-{3-[2-Ethyl-5-hydroxy-4-(1H-pyrazol-3-yl)-phe...)
Affinity DataIC50:  834nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50039474(3-(3-{3-[4-(1H-Pyrazol-3-yl)-phenoxy]-propoxy}-phe...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [3H]-Leukotriene B4 binding to human PMNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045094(7-(2-Carboxy-ethyl)-6-decyloxy-9-oxo-9H-xanthene-4...)
Affinity DataIC50:  1.77E+3nMAssay Description:Inhibition of specific binding of LTB4 ( 0.1 nM) to receptors on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50045095(5-(2-Carboxy-ethyl)-6-decyloxy-9-oxo-9H-xanthene-4...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of specific binding of LTB4 ( 0.1 nM) to receptors on intact human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed