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Found 1338 with Last Name = 'campobasso' and Initial = 'n'
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50159507(CHEMBL3785703)
Affinity DataKi:  0.800nMAssay Description:Competitive inhibition of human RIP1 (1 to 375 residues) in presence of increasing ATP by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92766(PDF inhibitor, compound 8)
Affinity DataKi:  53.7nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Escherichia coli)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50535516(CHEMBL4542964)
Affinity DataKi:  60nMAssay Description:Inhibition of Escherichia coli PDFMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92761(PDF inhibitor, compound 3)
Affinity DataKi:  117nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92764(PDF inhibitor, compound 6)
Affinity DataKi:  213nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92760(PDF inhibitor, compound 2)
Affinity DataKi:  334nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92765(PDF inhibitor, compound 7)
Affinity DataKi:  650nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169013(CHEMBL3805703)
Affinity DataKi:  2.90E+3nMAssay Description:Competitive inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) assessed as formation of G6P by continuou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92759(PDF inhibitor, compound 1)
Affinity DataKi:  6.31E+3nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92762(PDF inhibitor, compound 4)
Affinity DataKi:  2.59E+4nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Glaxosmithkline

LigandPNGBDBM92763(PDF inhibitor, compound 5)
Affinity DataKi:  3.17E+4nMAssay Description:Binding assay using PDF inhibitors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233227(CHEMBL4067372)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50159697(CHEMBL3785745)
Affinity DataIC50:  0.0630nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233256(CHEMBL4093220)
Affinity DataIC50:  0.0790nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383996(CHEMBL2032134)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383999(CHEMBL2032137)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383966(CHEMBL2032148)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383998(CHEMBL2032136)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50384000(CHEMBL2032138)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383997(CHEMBL2032135)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50159696(CHEMBL3786997)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50159696(CHEMBL3786997)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Flag-tagged human RIP1 (1 to 324 residues) after 30 mins by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383994(CHEMBL2032132)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383987(CHEMBL2032125)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383982(CHEMBL2032119)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383988(CHEMBL2032126)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383995(CHEMBL2032133)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383993(CHEMBL2032131)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233248(CHEMBL4096224)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233244(CHEMBL4068954)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383968(CHEMBL2032140)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50384003(CHEMBL2032142)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50384002(CHEMBL2032141)
Affinity DataIC50:  0.370nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383972(CHEMBL2032146)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50159693(CHEMBL3785482)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Flag-tagged human RIP1 (1 to 324 residues) after 30 mins by ADP-Glo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233255(CHEMBL4069318)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233225(CHEMBL4071864)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of RIP1 in human primary neutrophils assessed as reduction in TNFalpha/QCD-OPh/SMAC mimetic RMT 5265-induced necroptosis at 21 hrs post-st...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233228(CHEMBL4060644)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383969(CHEMBL2032143)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383980(CHEMBL2032117)
Affinity DataIC50:  0.430nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383992(CHEMBL2032130)
Affinity DataIC50:  0.440nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383965(CHEMBL2032129)
Affinity DataIC50:  0.460nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383967(CHEMBL2032122)
Affinity DataIC50:  0.480nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50513015(CHEMBL4537171)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human GST/His-tagged RIP1 (1 to 375 residues) expressed in baculovirus expression system assessed as reduction in autophosphorylation m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383981(CHEMBL2032118)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233226(CHEMBL4089558)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233230(CHEMBL4099004)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human RIP1 (1 to 375 residues) expressed in baculovirus infected insect cells preincubated for 1 hr followed by ATP addition measured a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50233225(CHEMBL4071864)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of RIP1 in human primary neutrophils assessed as reduction in TNFalpha/QCD-OPh/SMAC mimetic RMT 5265-MIP-1beta production at 21 hrs post-s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae serotype 4 (strain ATCC B...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383986(CHEMBL2032124)
Affinity DataIC50:  0.510nMAssay Description:Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383996(CHEMBL2032134)
Affinity DataIC50:  0.520nMAssay Description:Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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