TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Shinshu University
Curated by PDSP Ki Database
Shinshu University
Curated by PDSP Ki Database
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Shinshu University
Curated by PDSP Ki Database
Shinshu University
Curated by PDSP Ki Database
Affinity DataKi: 0.770nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]-DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]-DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Shinshu University
Curated by PDSP Ki Database
Shinshu University
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]-DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]-DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]-DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]-DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Binding affinities against Opioid receptor delta 1 of guinea pig brain membrane using [3H]-DPDPE as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataKi: 1.55E+3nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
Affinity DataIC50: 0.00700nMAssay Description:Binding affinities against Opioid receptor mu 1 of guinea pig brain membrane using [3H]-DAGO as the radioligand using competition binding assays.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of VLA-4 to VCAM-1 bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a protein-based ligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Evaluated for inhibitory activity against Opioid receptor mu 1 of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of binding of Very late antigen 4/vascular cell adhesion molecule 1 in a protein-based ligand binding assayMore data for this Ligand-Target Pair