Affinity DataKi: 0.00140nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.00150nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0150nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0170nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0180nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0190nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0210nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0210nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0220nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0330nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0340nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0420nMAssay Description:Inhibitory constant against thrombin (IIa) More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0450nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0460nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0560nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0850nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0870nMAssay Description:Inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.0940nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0960nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity towards thrombin was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory constant against thrombin (IIa) More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Merck Research Labortories
Curated by ChEMBL
Merck Research Labortories
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Displacement of [125I]-hCGRP from human CGRP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Compound was evaluated to inhibit the thrombin enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.125nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibitory constant against thrombin (IIa) More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Binding affinity of the compound was evaluated on serine protease thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity towards thrombin was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Inhibitory activity of the compound against thrombin (IIa) was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibitory constant against thrombin (IIa) More data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Binding affinity to human bradikinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibitory potency against human thrombinMore data for this Ligand-Target Pair