Affinity DataKi: 0.220nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.720nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.980nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibitory Activity against bovine thrombinMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 6.80nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 7.10nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of human thymidylate synthase expressed in Escherichia coli incubated for 1 hr by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibitory Activity against bovine alpha-thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Serotonergic activity of the compound.More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibitory Activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Kinetic inhibition constant evaluated by measuring serotonergic activityMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair