Compile Data Set for Download or QSAR
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Found 16 with Last Name = 'derrien' and Initial = 'm'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281664(CHEMBL262894 | p-Tyr(SO3Na)-gNle-mGly-Trp-(N-Me)Nl...)
Affinity DataKi:  0.0600nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50016504((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...)
Affinity DataKi:  0.150nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281665(Boc-Phe(CH2-SO3Na)-gNle-mCIy-Trp-(N-Me)Nle-Asp-Phe...)
Affinity DataKi:  0.460nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.640nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.640nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  11nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Merk CCK-B antagonist L365,260 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  14nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281666(Boc-Trp-Phg-Asp-1Nal-N(CH3)2 | CHEMBL436722)
Affinity DataKi:  39nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  51nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type B receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281664(CHEMBL262894 | p-Tyr(SO3Na)-gNle-mGly-Trp-(N-Me)Nl...)
Affinity DataKi:  62nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281668(Boc-Trp-Phe-Asp-1Nal-NH2 | CHEMBL171594)
Affinity DataKi:  71nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 to Cholecystokinin type B receptor in guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50016504((S)-3-(2-{[(S)-2-(2-{2-[2-tert-Butoxycarbonylamino...)
Affinity DataKi:  78nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281666(Boc-Trp-Phg-Asp-1Nal-N(CH3)2 | CHEMBL436722)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281669(Boc-Trp-Phg-Asp-1Nal-NH2 | CHEMBL353862)
Affinity DataKi:  1.10E+3nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281665(Boc-Phe(CH2-SO3Na)-gNle-mCIy-Trp-(N-Me)Nle-Asp-Phe...)
Affinity DataKi:  1.10E+3nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281668(Boc-Trp-Phe-Asp-1Nal-NH2 | CHEMBL171594)
Affinity DataKi:  2.40E+3nMAssay Description:Tested for the inhibition of [3H]-pCCK-8 binding to Cholecystokinin type A receptor in pancreatic membranes of guinea-pigMore data for this Ligand-Target Pair
In DepthDetails Article