Compile Data Set for Download or QSAR
maximum 50k data
Found 470 with Last Name = 'ernst' and Initial = 'b'
TargetSialidase-4(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50270464(CHEMBL4076203)
Affinity DataKi:  260nMAssay Description:Inhibition of human N-terminal MBP-fused NEU4 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-3(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50270464(CHEMBL4076203)
Affinity DataKi:  280nMAssay Description:Inhibition of human N-terminal MBP-fused NEU3 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-3(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50270441(CHEMBL4099818)
Affinity DataKi:  320nMAssay Description:Inhibition of human N-terminal MBP-fused NEU3 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-3(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataKi:  620nMAssay Description:Inhibition of human N-terminal MBP-fused NEU3 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-3(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human N-terminal MBP-fused NEU3 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-4(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50270441(CHEMBL4099818)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human N-terminal MBP-fused NEU4 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataKi:  5.70E+3nMAssay Description:Inhibition of human N-terminal MBP-fused NEU2 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetSialidase-4(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataKi:  5.80E+3nMAssay Description:Inhibition of human N-terminal MBP-fused NEU4 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50270441(CHEMBL4099818)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of human N-terminal MBP-fused NEU2 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM4706((2R,3R,4S)-3-acetamido-4-hydroxy-2-[(1R,2R)-1,2,3-...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of human N-terminal MBP-fused NEU2 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
TargetSialidase-4(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataKi:  2.60E+4nMAssay Description:Inhibition of human N-terminal MBP-fused NEU4 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50270464(CHEMBL4076203)
Affinity DataKi:  4.80E+4nMAssay Description:Inhibition of human N-terminal MBP-fused NEU2 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM26258((1S,2R,9R,10R,11S,14S,15S)-14-hydroxy-9,14,15-trim...)
Affinity DataIC50:  1.66nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50:  2nMAssay Description:Inhibition of ATR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410541(CHEMBL194467)
Affinity DataIC50:  2.24nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410489(TRENBOLONE)
Affinity DataIC50:  2.63nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50367916(METHYLTRIENOLONE | Metribolone | R-1881)
Affinity DataIC50:  3.09nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347464(CHEMBL1802187)
Affinity DataIC50:  4.80nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347465(CHEMBL1802185)
Affinity DataIC50:  6.70nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354062(CHEMBL1836190)
Affinity DataIC50:  9nMAssay Description:Inhibition of MAG -Fc chimera expressed in CHO cells using NeuAc alpha2-3Galbeta1-4GlcNAc-R coupled biotinylated polyacrylamide after 30 mins by ELIS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347449(CHEMBL1171278)
Affinity DataIC50:  10.4nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410518(CHEMBL371356)
Affinity DataIC50:  11.0nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347450(CHEMBL1802194)
Affinity DataIC50:  11.8nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347451(CHEMBL1802191)
Affinity DataIC50:  15.3nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410531(Android | Android 10 | Android 25 | Android 5 | ME...)
Affinity DataIC50:  15.8nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410492(EPITESTOSTERONE)
Affinity DataIC50:  15.8nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347452(CHEMBL1802190)
Affinity DataIC50:  16nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347453(CHEMBL1802186)
Affinity DataIC50:  17.1nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410522(LEVONORGESTREL)
Affinity DataIC50:  19nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347454(CHEMBL1171678)
Affinity DataIC50:  20nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347455(CHEMBL1802188)
Affinity DataIC50:  22nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347456(CHEMBL1802192)
Affinity DataIC50:  23.9nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347457(CHEMBL1802189)
Affinity DataIC50:  27.6nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347458(CHEMBL1802195)
Affinity DataIC50:  29.2nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347459(CHEMBL1802193)
Affinity DataIC50:  38.7nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataIC50:  65.6nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357403(CHEMBL1917312)
Affinity DataIC50:  70nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347460(CHEMBL1170455)
Affinity DataIC50:  73nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyelin-associated glycoprotein(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50354056(CHEMBL1836336)
Affinity DataIC50:  79nMAssay Description:Inhibition of MAG -Fc chimera expressed in CHO cells using NeuAc alpha2-3Galbeta1-4GlcNAc-R coupled biotinylated polyacrylamide after 30 mins by ELIS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410516(CHEMBL263818)
Affinity DataIC50:  89.1nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50405375(CHEMBL194749)
Affinity DataIC50:  89.1nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357424(CHEMBL1917473)
Affinity DataIC50:  112nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50148732(17-ethynyl-17beta-hydroxyestr-4-en-3-one | 17alpha...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50410527(CHEMBL194858)
Affinity DataIC50:  135nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357407(CHEMBL1917308)
Affinity DataIC50:  135nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357418(CHEMBL1917479)
Affinity DataIC50:  144nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM36025(phenyl-beta-d-glucopyranoside)
Affinity DataIC50:  150nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357423(CHEMBL1917474)
Affinity DataIC50:  153nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357426(CHEMBL1917471)
Affinity DataIC50:  161nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50357410(CHEMBL1917305)
Affinity DataIC50:  169nMAssay Description:Antagonist activity at Escherichia coli recombinant C-terminal 6His-tagged FimH-CRD with a C-terminal thrombin cleavage site expressed in Escherichia...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 470 total ) | Next | Last >>
Jump to: