TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 0.302nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 0.650nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 0.760nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.870nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity towards alpha-2a adrenergic receptorMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University Of Tennessee-Memphis
Curated by ChEMBL
University Of Tennessee-Memphis
Curated by ChEMBL
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
Affinity DataKi: 2.80nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Ohio State University
Curated by PDSP Ki Database
Ohio State University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair