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Found 303 with Last Name = 'fornaretto' and Initial = 'mg'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033857(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  0.5nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033857(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  0.5nMAssay Description:Binding affinity against serotonin 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033852(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  0.540nMAssay Description:Binding affinity against serotonin 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033852(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  0.540nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289537(1-(3-Phenyl-propyl)-3-((Z)-styryl)-piperidine | CH...)
Affinity DataIC50:  0.600nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  0.770nMAssay Description:Binding affinity against serotonin 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  0.770nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289553(1-Phenethyl-3-((Z)-styryl)-piperidine | CHEMBL3697...)
Affinity DataIC50:  0.800nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289552(1-(3-Methyl-but-2-enyl)-3-((Z)-styryl)-piperidine ...)
Affinity DataIC50:  1nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033835(1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  1.70nMAssay Description:Binding affinity against serotonin 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070198((6aR,9R,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,9,1...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289539(1-Cyclohexyl-3-((Z)-styryl)-piperidine | CHEMBL398...)
Affinity DataIC50:  2nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataIC50:  2.10nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataIC50:  2.10nMAssay Description:Binding affinity against serotonin 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070192((6aR,9R,10aR)-3-tert-Butyl-7-methyl-4,6,6a,7,8,9,1...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070187(1-Acetyl-3-((6aR,9S,10aR)-3-tert-butyl-7-methyl-4,...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H...)
Affinity DataIC50:  3.40nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 2A receptor was evaluated using [3H]- ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054990(1-[2-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataIC50:  3.60nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054999(1-[2-(6-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl...)
Affinity DataIC50:  3.70nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289538(1-Allyl-3-((E)-styryl)-piperidine | CHEMBL39735)
Affinity DataIC50:  4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289541(1-(3-Phenyl-propyl)-3-((E)-styryl)-piperidine | CH...)
Affinity DataIC50:  4nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50:  4.80nMAssay Description:Affinity towards Dopamine receptor D2 was evaluated in rat striatal membrane using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50:  4.80nMAssay Description:Binding affinity to rat Dopamine receptor D2 expressed in CHO cells was determined using [125 I ] iodosulpride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataIC50:  5.20nMAssay Description:Binding affinity towards rat Dopamine receptor D2 was evaluated using [3H]- spiroperidol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataIC50:  5.20nMAssay Description:Binding affinity to rat Dopamine receptor D2 expressed in CHO cells was determined using [125 I ] iodosulpride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054997(1-[3-(6-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  5.40nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289549(1-Cyclohexyl-3-((E)-styryl)-piperidine | CHEMBL291...)
Affinity DataIC50:  6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289547(1-Phenethyl-3-((E)-styryl)-piperidine | CHEMBL2879...)
Affinity DataIC50:  6nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50070193(1-((6aR,9R,10aR)-2-tert-Butyl-7-methyl-4,6,6a,7,8,...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]yohimbine from Alpha-2 adrenergic receptor in rat frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289551(1-(4-Phenyl-butyl)-3-((Z)-styryl)-piperidine | CHE...)
Affinity DataIC50:  7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50289545(1-(2-Cyclohexyl-ethyl)-3-((Z)-styryl)-piperidine |...)
Affinity DataIC50:  7nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054989(1-[2-(7-Methoxy-3,4-dihydro-naphthalen-2-yl)-ethyl...)
Affinity DataIC50:  7.30nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033847(CHEMBL108241 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  7.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054996(1-[2-(6-Methoxy-3,4-dihydro-naphthalen-2-yl)-ethyl...)
Affinity DataIC50:  8.20nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50052561(CHEMBL326017 | {2-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  8.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033854(1-[3-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  9.20nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50052569(CHEMBL107486 | {3-[4-(2-Methoxy-phenyl)-piperazin-...)
Affinity DataIC50:  10nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampus membranes using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289536(1-Benzyl-3-((E)-styryl)-piperidine | CHEMBL39855)
Affinity DataIC50:  10nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054991(1-[2-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  12nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 2A receptor was evaluated using [3H]- ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289554(1-Pent-4-enyl-3-((E)-styryl)-piperidine | CHEMBL38...)
Affinity DataIC50:  12nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50070203(CHEMBL14048 | N-((6aR,9S,10aR)-7-Methyl-4,6,6a,7,8...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50070201(((6aR,9S,10aR)-2-tert-Butyl-7-methyl-4,6,6a,7,8,9,...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289540(1-(3-Phenoxy-propyl)-3-((Z)-styryl)-piperidine | C...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50054998(1-[4-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50:  15nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033835(1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  15nMAssay Description:Binding affinity against Dopamine receptor D2 in rat striatal membrane using [3H]spiroperidol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50289544(1-Phenyl-4-[3-((Z)-styryl)-piperidin-1-yl]-butan-1...)
Affinity DataIC50:  15nMAssay Description:Binding affinity at sigma receptor by [3H]-(+)-SKF-10,047 displacement.More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50052565(5-Methoxy-1,2,3,4-tetrahydro-naphthalene-1-carboxy...)
Affinity DataIC50:  16nMAssay Description:Binding affinity against serotonin 5-hydroxytryptamine 1A receptor in rat hippocampus membrane using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033850(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50:  18nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 1A receptor was evaluated using [3H]8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  18nMAssay Description:Binding affinity towards rat Dopamine receptor D2 was evaluated using [3H]- spiroperidol as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50:  18nMAssay Description:Binding affinity to rat Dopamine receptor D2 expressed in CHO cells was determined using [125 I ] iodosulpride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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