Affinity DataKi: 0.100nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHO-D cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHOD cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity to cannabinoid CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Binding affinity to cannabinoid CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]Lys-desArg9-BK from human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity to mouse EP4 receptor by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHOD cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHO-D cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.851nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.09nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Binding affinity to human recombinant 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHO-D cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHO-D cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.98nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.2 T: 2°CAssay Description:Enzyme assays were performed using purified recombinant human or mouse11beta-HSD1. The fractional conversion of cortisone to cortisol was used to det...More data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.2 T: 2°CAssay Description:The 11beta-HSD1 enzyme assay was carried out in the replica plates of the compounds in reaction buffer containing substrate mixture [3H]-cortisone/NA...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]Lys-desArg9-BK from human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity to cannabinoid CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]Lys-desArg9-BK from human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]Lys-desArg9-BK from human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]DAK from human bradykinin B1 receptor expressed in CHOD cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.5kJ/molepH: 7.2 T: 2°CAssay Description:Enzyme assays were performed using purified recombinant human or mouse11beta-HSD1. The fractional conversion of cortisone to cortisol was used to det...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Antagonist activity at human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]Lys-desArg9-BK from human bradykinin B1 receptorMore data for this Ligand-Target Pair