TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 0.339nM ΔG°: -54.1kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.407nM ΔG°: -53.6kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 0.794nMAssay Description:In vitro affinity for muscarinic M3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -51.4kJ/mole EC50: 2nMpH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro affinity for muscarinic M3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
UniversitÉ
Curated by PDSP Ki Database
UniversitÉ
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]N-methylscopolamine from human recombinant M3 muscarinic receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro affinity for muscarinic M3 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Antagonism of Muscarinic M3 receptors as displacement of concentration response curve of carbachol on isolated guinea-pig urinary bladderMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nM ΔG°: -49.7kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Muscarinic M3 receptors as displacement of concentration response curve of carbachol on isolated guinea-pig urinary bladderMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Muscarinic M3 receptors as displacement of concentration response curve of carbachol on isolated guinea-pig urinary bladderMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Antagonism of Muscarinic M3 receptors as displacement of concentration response curve of carbachol on isolated guinea-pig ileumMore data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.6kJ/molepH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH3R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]methylscopolamine from recombinant human muscarinic M3 receptors expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]-substance P from human NK1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]N-methylscopolamine from human recombinant M3 muscarinic receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair