Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of alpha1B adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Inhibition of alpha1B adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of BACE1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 128nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 174nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 179nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 217nMAssay Description:Inhibition of CA-9 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Regina Elena National Cancer Institute
Curated by ChEMBL
Regina Elena National Cancer Institute
Curated by ChEMBL
Affinity DataIC50: 223nMAssay Description:Displacement of [3H]R-1881 from Androgen receptor of PC3-AR cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 226nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 248nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 255nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 266nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 295nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.62E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.32E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.07E+3nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.44E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.57E+3nMAssay Description:Inhibition of CA-12 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-1 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CA-2 (unknown origin) after 15 mins by CO2 hydration assayMore data for this Ligand-Target Pair
TargetBile acid receptor(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataEC50: >3.16E+4nMAssay Description:Agonist activity at human FXR expressed in COS1 cells by luciferase assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Centre National de la Recherche Scientifique/INSERM/ULP
Curated by ChEMBL
Affinity DataEC50: 2.18E+3nMAssay Description:Agonist activity at human TGR5 expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair