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Found 741 with Last Name = 'giordani' and Initial = 'a'
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50435130(CHEMBL1893324)
Affinity DataKi:  0.0670nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50015490(CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITR...)
Affinity DataKi:  0.0760nMAssay Description:Binding affinity to human neuropeptide Y receptor type 2 by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50015490(CHEMBL438945 | H-YPSKPDNPGEDAPAEDMARYYSALRHYINLITR...)
Affinity DataKi:  0.0960nMAssay Description:Binding affinity to human neuropeptide Y receptor type 1 by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50335566(CHEMBL1651026 | Substance P [Sar9,Met(O2)11])
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human NK1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007158((S)-2-(3,4-Dichloro-phenyl)-1-(2-pyrrolidin-1-ylme...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50130880(CHEMBL407196 | NT(1-13) | neurotensin | pGlu-Leu-T...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to human NTS1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008888((threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-methyl-pyrr...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008888((threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-methyl-pyrr...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50333104(CHEMBL389521 | H-FGGFTGARKSARKLANQ-NH2 | N/OFQ-NH2...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity to human NOP receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000278(2-(3,4-Dichloro-phenyl)-1-(2-piperidin-1-ylmethyl-...)
Affinity DataKi:  0.480nMAssay Description:Compound was evaluated for its binding affinity against Opioid receptor kappa 1 subtype in guinea pig brain (minus cerebellum)using [3H]-U-69,593 as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000287(2-(3,4-Dichloro-phenyl)-1-(2-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  0.530nMAssay Description:Compound was evaluated for its binding affinity against Opioid receptor kappa 1 subtype in guinea pig brain (minus cerebellum) .using [3H]-U-69,593 a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008895(1-(2-Pyrrolidin-1-ylmethyl-piperidin-1-yl)-2-(4-tr...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008895(1-(2-Pyrrolidin-1-ylmethyl-piperidin-1-yl)-2-(4-tr...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50452995(CHEMBL2111856)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50366495((+)butaclamol | CHEMBL1255588)
Affinity DataKi:  0.740nMAssay Description:Binding affinity to human dopamine D2S receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008897(2-(4-Bromo-phenyl)-1-(2-pyrrolidin-1-ylmethyl-pipe...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)
Affinity DataKi:  0.950nMAssay Description:Binding affinity to human histamine H1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008898(1-(2-Pyrrolidin-1-ylmethyl-piperidin-1-yl)-2-(3-tr...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008899(2-(3,4-Dichloro-phenyl)-1-(2-diethylaminomethyl-pi...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000267(2-(3,4-Dichloro-phenyl)-1-(2-dimethylaminomethyl-p...)
Affinity DataKi:  1.40nMAssay Description:Compound was evaluated for its binding affinity against Opioid receptor kappa 1 subtype in guinea pig brain (minus cerebellum)using [3H]-U-69,593 as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to human glucocorticoid receptor by radioligand displacement assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008892(2-(4-Chloro-phenyl)-1-(2-pyrrolidin-1-ylmethyl-pip...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008893(2-(3,4-Dimethyl-phenyl)-1-(2-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human GAL2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]-DAGO from mu opioid receptors in guinea pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50051295((S)-3-methyl-2-phenyl-N-(1-phenylpropyl)quinoline-...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human NK3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008894(1-(2-Pyrrolidin-1-ylmethyl-piperidin-1-yl)-2-p-tol...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM82561(CAS_40796-97-2 | TROPANYL 3,5-DICHLOROBENZOATE | T...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity to human 5-HT3 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM23954(5-[(2E,3aS,4R,5R,6aS)-5-hydroxy-4-[(1E,3S)-3-hydro...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human PGI2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50435131(CHEMBL2390989)
Affinity DataKi:  5nMAssay Description:Binding affinity to human NK2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50435129(CHEMBL2392354)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to human bradykinin B2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008896(1-(2-Pyrrolidin-1-ylmethyl-piperidin-1-yl)-2-(2-tr...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50119657(8-Butyl-7-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008891(2-(4-Fluoro-phenyl)-1-(2-pyrrolidin-1-ylmethyl-pip...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50452994(CHEMBL2111857)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50089990(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Universit£

Curated by ChEMBL
LigandPNGBDBM50119658(7-Butyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataKi:  140nMAssay Description:Binding affinity to human histamine H2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008890(2-(4-Hydroxy-phenyl)-1-(2-pyrrolidin-1-ylmethyl-pi...)
Affinity DataKi:  194nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  460nMAssay Description:Compound was evaluated for its binding affinity against opioid receptor delta subtype in guinea pig brain (minus cerebellum)using [3H]-DADLE as radio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008888((threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-methyl-pyrr...)
Affinity DataKi:  464nMAssay Description:Displacement of [3H]-DAGO from mu opioid receptors in guinea pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008888((threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-methyl-pyrr...)
Affinity DataKi:  464nMAssay Description:Displacement of [3H]-DAGO from mu opioid receptors in guinea pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50000296(CHEMBL441765 | CHEMBL482811 | U-50488H | US1149237...)
Affinity DataKi:  616nMAssay Description:Displacement of [3H]-DAGO from mu opioid receptors in guinea pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008889((threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-dimethylami...)
Affinity DataKi:  762nMAssay Description:Displacement of [3H]-DAGO from mu opioid receptors in guinea pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008900(2-(4-Cyclohexyl-phenyl)-1-(2-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  827nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008900(2-(4-Cyclohexyl-phenyl)-1-(2-pyrrolidin-1-ylmethyl...)
Affinity DataKi:  974nMAssay Description:Displacement of [3H]-DAGO from mu opioid receptors in guinea pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50008889((threo)2-(3,4-Dichloro-phenyl)-1-[2-(1-dimethylami...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-U-69,593 from kappa opioid receptors in guine pig brain (minus cerebellum).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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