Affinity DataKi: 0.0570nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0640nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 0.0770nMAssay Description:Compound was evaluated for its affinity for Alpha-1a adrenergic receptor in human aorta preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0840nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 0.0990nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Compound was evaluated for its affinity for alpha 1a receptor in human prostate tissue preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Compound was evaluated for its affinity for Alpha-1a adrenergic receptor in human prostate tissue preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor using 0.1 nM [3H]-8-OH-DPAT (8-hydroxy-2-(di-n-propylamino)tet-ralin), from rat hippocampal ...More data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human Alpha-1a adrenergic receptor stably expressed in Chinese...More data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Compound was tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1b adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding activity against alpha-2 adrenergic receptor from calf cerebral cortex, using [3H]-clonidine as the radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Compound was tested for inhibition of hog kidney reninMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl) ethylamino methyl tetralone from human cloned Alpha-1d adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Compound was evaluated for its affinity for Alpha-1a adrenergic receptor in human aorta preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Compound was evaluated for its affinity for Alpha-1a adrenergic receptor in human aorta preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding activity against alpha-2 adrenergic receptor from calf cerebral cortex, using [3H]-clonidine as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding activity against alpha-2 adrenergic receptor from calf cerebral cortex, using [3H]-clonidine as the radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylaminomethyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in ...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1b adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Ability to displace beta ([125I]-iodo-4-hydroxyphenyl)-ethylamino methyl tetralone from human cloned Alpha-1a adrenergic receptor stably expressed in...More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity for rat oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity for rat oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity for cloned human oxytocin receptor (OT-R)More data for this Ligand-Target Pair