Affinity DataIC50: 0.5nMAssay Description:Compound was tested for its inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory potency on plasma renin obtained from catsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory potency on plasma renin obtained from mongrel dogsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Compound was tested for its inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory potency on plasma renin obtained from mongrel dogsMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory potency on plasma renin obtained from hypertensive humansMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory potency on plasma renin obtained from mongrel dogsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Compound was tested for its inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Compound was tested for its inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibitory potency on plasma renin obtained from hypertensive humansMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory potency on plasma renin obtained from hypertensive humansMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibitory potency on plasma renin obtained from catsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory potency on plasma renin obtained from New Zealand white rabbitsMore data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Eberhard Karls University Tuebingen
Curated by ChEMBL
Eberhard Karls University Tuebingen
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of mPGES1 in IL1beta induced human A549 cell microsomal membrane assessed as blockade of conversion of PGH2 to PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibitory potency on plasma renin obtained from hypertensive humansMore data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Eberhard Karls University Tuebingen
Curated by ChEMBL
Eberhard Karls University Tuebingen
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of mPGES1 in IL1beta induced human A549 cell microsomal membrane assessed as blockade of conversion of PGH2 to PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 280nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair