Affinity DataKi: 0.00300nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity to dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity to human CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity to human CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity to human CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 0.980nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 1.25nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]CP55940 from CB1 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 1.49nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 1.65nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 1.92nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 2.23nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Tours
Curated by PDSP Ki Database
University Of Tours
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 2.75nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Karolinska Institutet
Curated by PDSP Ki Database
Karolinska Institutet
Curated by PDSP Ki Database
Affinity DataKi: 5.80nMAssay Description:Inhibition of [3H]-nisoxatine binding to norepinephrine transporter (NET) of rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 7.93nMAssay Description:Binding affinity at NETMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 7.96nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.29nMAssay Description:Binding affinity at NETMore data for this Ligand-Target Pair
Affinity DataKi: 10.8nMAssay Description:Binding affinity at NETMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Tours
Curated by PDSP Ki Database
University Of Tours
Curated by PDSP Ki Database
Affinity DataKi: 12nMAssay Description:Displacement of [125I]PE2I from rat DATMore data for this Ligand-Target Pair
Affinity DataKi: 12.8nMAssay Description:Inhibition of [3H]-nisoxatine binding to norepinephrine transporter (NET) of rat cortical homogenatesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 15.7nMAssay Description:Displacement of [3H]CP55940 from CB1 receptorMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Tours
Curated by PDSP Ki Database
University Of Tours
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Displacement of [125I]PE2I from rat DATMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 16.9nMAssay Description:Binding affinity to human CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 17.4nMAssay Description:Binding affinity to human CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Tours
Curated by PDSP Ki Database
University Of Tours
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 19.3nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 28.4nMAssay Description:Inhibition of [3H]-nisoxatine binding to norepinephrine transporter (NET) of rat cortical homogenatesMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Karolinska Institutet
Curated by PDSP Ki Database
Karolinska Institutet
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours
Curated by ChEMBL
University Of Tours
Curated by ChEMBL
Affinity DataKi: 53.3nMAssay Description:Inhibition of [3H]-paroxetine binding to serotonin transporter (SERT) of rat cortical membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]CP55940 from CB1 receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 61.8nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 62.2nMAssay Description:Displacement of [3H]CP55940 from CB1 receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 75.2nMAssay Description:Displacement of [3H]PK11195 from TSPO receptor in rat kidney membranesMore data for this Ligand-Target Pair
Affinity DataKi: 80.2nMAssay Description:Inhibition of [3H]-nisoxatine binding to norepinephrine transporter (NET) of rat cortical homogenatesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor at 10 uM by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Inhibition of [3H]-nisoxatine binding to norepinephrine transporter (NET) of rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 107nMAssay Description:Inhibition of [3H]-nisoxatine binding to norepinephrine transporter (NET) of rat cortical homogenatesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 115nMAssay Description:Displacement of [3H]CP55940 from CB1 receptorMore data for this Ligand-Target Pair