Compile Data Set for Download or QSAR
maximum 50k data
Found 27 with Last Name = 'hopson' and Initial = 'j'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265490(CHEMBL501238 | N-{m-[R(+)-1]Ureaphenoxy}ethyldigly...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]DAMGO from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265491(1-{1-Diglycoldiamide-2-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265491(1-{1-Diglycoldiamide-2-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]DAMGO from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265490(CHEMBL501238 | N-{m-[R(+)-1]Ureaphenoxy}ethyldigly...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DAMGO from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265493(CHEMBL442943 | N-{m-[R(+)-1]Ureaphenoxy}ethyl-N'-o...)
Affinity DataKi:  14.2nMAssay Description:Displacement of [3H]DAMGO from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265492(1-{1-Diglycoldiamide-6-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  16.3nMAssay Description:Displacement of [3H]DAMGO from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265494((R)-N-methyl-2-(1-(3-(3-(1-methyl-2-oxo-5-phenyl-2...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265493(CHEMBL442943 | N-{m-[R(+)-1]Ureaphenoxy}ethyl-N'-o...)
Affinity DataKi:  24.1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265492(1-{1-Diglycoldiamide-6-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  29.4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265533(2-({[(1S,5R,13R,14S,17S)-9,17-dihydroxy-4-methyl-1...)
Affinity DataKi:  29.8nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265491(1-{1-Diglycoldiamide-2-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  33nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265533(2-({[(1S,5R,13R,14S,17S)-9,17-dihydroxy-4-methyl-1...)
Affinity DataKi:  40.7nMAssay Description:Displacement of [3H]DAMGO from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265494((R)-N-methyl-2-(1-(3-(3-(1-methyl-2-oxo-5-phenyl-2...)
Affinity DataKi:  48nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265490(CHEMBL501238 | N-{m-[R(+)-1]Ureaphenoxy}ethyldigly...)
Affinity DataKi:  57nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265491(1-{1-Diglycoldiamide-2-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  71nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265492(1-{1-Diglycoldiamide-6-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  77nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265493(CHEMBL442943 | N-{m-[R(+)-1]Ureaphenoxy}ethyl-N'-o...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2R-MOPR (unknown origin) coexpressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265493(CHEMBL442943 | N-{m-[R(+)-1]Ureaphenoxy}ethyl-N'-o...)
Affinity DataKi:  223nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265492(1-{1-Diglycoldiamide-6-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataKi:  260nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265490(CHEMBL501238 | N-{m-[R(+)-1]Ureaphenoxy}ethyldigly...)
Affinity DataKi:  356nMAssay Description:Displacement of [125I]CCK-26-33 from CCK2 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265491(1-{1-Diglycoldiamide-2-[m-(R(+)-1)ureaphenoxy]etha...)
Affinity DataEC50:  119nMAssay Description:Activity at CCK2R-MOPR (unknown origin) coexpressed in CHO cells cotransfected with delta6-Galphaqi4-myr assessed as intracellular calcium release by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataEC50:  2.66nMAssay Description:Activity at CCK2R-MOPR (unknown origin) coexpressed in CHO cells cotransfected with delta6-Galphaqi4-myr assessed as intracellular calcium release by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50265533(2-({[(1S,5R,13R,14S,17S)-9,17-dihydroxy-4-methyl-1...)
Affinity DataEC50:  572nMAssay Description:Activity at CCK2R-MOPR (unknown origin) coexpressed in CHO cells cotransfected with delta6-Galphaqi4-myr assessed as intracellular calcium release by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed