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Found 82 with Last Name = 'ireland' and Initial = 'sj'
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007824(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50: >3.57E+3nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007823(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propionyla...)
Affinity DataEC50:  188nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007825(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  130nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007825(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007826(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007827(2-(3-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007828(2-(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007828(2-(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50: >500nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007829(2-(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007823(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propionyla...)
Affinity DataEC50:  188nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007830(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propionyla...)
Affinity DataEC50:  400nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007831(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007822(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  892nMAssay Description:Agonistic activity at neurokinin-1 (NK-1) receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007830(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propionyla...)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  1nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007831(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  6.90nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007826(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  1.20nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007832(2-(3-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007832(2-(3-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007822(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50: >100nMAssay Description:Agonist activity was measured at neurokinin-2 receptor in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007827(2-(3-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  15nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007829(2-(1-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50:  63nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50007824(2-(2-{2-[2-(4-Amino-butyrylamino)-3-phenyl-propion...)
Affinity DataEC50: >300nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001603(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  307nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001593(CHEMBL131872 | N-{1-[1-(1-{1-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  4.24E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001594(CHEMBL335054 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  61nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001602(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  3.73E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001606(2-(2-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001595(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50:  13nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001607(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50:  830nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001604(2-(2-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  38nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001600(CHEMBL267712 | N-{1-[1-(1-Benzyl-2-{5-[1-(1-carbam...)
Affinity DataEC50:  1.03E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001447(CHEMBL217406 | His-Lys-Thr-Asp-Ser-Phe-Val-Gly-Leu...)
Affinity DataEC50:  14nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001596(3-(2-Acetylamino-6-amino-hexanoylamino)-N-{1-[1-(1...)
Affinity DataEC50:  44nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001598(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  5.23E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001592(CHEMBL131923 | N-{1-[1-(1-{5-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  1.13E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001599(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  545nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataEC50:  68nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataEC50:  5.60nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001601(2-(3-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001605(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50:  3.77E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001597(CHEMBL134481 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  45nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001592(CHEMBL131923 | N-{1-[1-(1-{5-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  59nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001593(CHEMBL131872 | N-{1-[1-(1-{1-[1-(1-Carbamoyl-3-met...)
Affinity DataEC50:  1.18E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001594(CHEMBL335054 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  870nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001595(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propiony...)
Affinity DataEC50:  1.30E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001596(3-(2-Acetylamino-6-amino-hexanoylamino)-N-{1-[1-(1...)
Affinity DataEC50:  1.30nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001597(CHEMBL134481 | N-(1-{1-[1-({[1-(1-Carbamoyl-3-meth...)
Affinity DataEC50:  33nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Glaxo Group Research

Curated by ChEMBL
LigandPNGBDBM50001599(2-(1-{2-[2-(5-Amino-pentanoylamino)-3-phenyl-propi...)
Affinity DataEC50: >1.80E+4nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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