Affinity DataKi: 0.0230nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Binding affinity towards Rabbit Coagulation factor X in a rabbit arterio-venous (A-V) shunt modelMore data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Binding affinity towards human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0370nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Binding affinity towards human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Binding affinity towards Rabbit Coagulation factor X in a rabbit arterio-venous (A-V) shunt modelMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 5(Macaca fascicularis)
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [125I]-MIP-1alpha from CCR5 in rhesus monkey Chem-1 cell membranes after 120 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity towards human trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Inhibition of matrix metalloprotease-13More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity imidazole glycerol phosphate dehydratase (IGPD) obtained from Cryptococcus neoformansMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity was evaluated against matrix metalloproteinase-1More data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]-naloxone from human mu opioid receptor expressed in CHO cells after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of matrix metalloprotease-7More data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:In vitro inhibition of human MMP-9.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated against matrix metalloproteinase-9More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-9.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-9.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-9.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-9.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-9.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:In vitro inhibition of human MMP-1.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity was evaluated against matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity was evaluated against matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity was evaluated against matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataKi: <1nMAssay Description:Binding affinity was evaluated against matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated against matrix metalloproteinase-9More data for this Ligand-Target Pair