TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Displacement of [3H]-5HT from human SERTMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 13.9nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 14.6nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 20.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 27.8nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]-5HT from human SERTMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 36.2nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 45.6nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 48.3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 51.7nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 53.8nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 71.6nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 76.1nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 76.7nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 83.5nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 101nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 115nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 116nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 124nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 184nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 203nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 221nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 222nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 274nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 275nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 711nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 719nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 777nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 944nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Medicines Institute
Curated by ChEMBL
National Medicines Institute
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in cerebral cortex homogenates after 15 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw
Curated by ChEMBL
Medical University Of Warsaw
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair