Affinity DataKi: 150nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement of [3H]R-PIA from adenosine A1 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 680nMAssay Description:Displacement of [3H]PSB-11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.13E+3nMAssay Description:Displacement of [3H]-MSX-2 from Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.18E+3nMAssay Description:Displacement of [3H]NECA from Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.26E+3nMAssay Description:Displacement of [3H]CCPA from Adenosine A1 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.94E+3nMAssay Description:Displacement of [3H]PSB-11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.20E+3nMAssay Description:Binding affinity towards human adenosine A2B receptor in VA13 fibroblasts as inhibition of adenylate cyclase at 10 uM; Less than 10% inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 9.45E+3nMAssay Description:Displacement of [3H]DPCPX from rat Adenosine A1 receptor of cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PSB-298 from human adenosine A2B receptor expressed in HEK293 cells at 10 uMMore data for this Ligand-Target Pair
Affinity DataKi: 1.39E+4nMAssay Description:Displacement of [3H]PSB-298 from human adenosine A2B receptor expressed in HEK293 cells at 10 uM; Less than 10% inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 1.71E+4nMAssay Description:Displacement of [3H]-MSX-2 from Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes without GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes with GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 680nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes without GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of human recombinant aromataseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of human leukocyte elastase using MeOSuc-Ala-Ala-Pro-Val-para-nitroanilide chromogenic substrate after 10 mins spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of forskolin-stimulated cAMP accumulation in chinese hamster ovary cell membranes expressing human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ptpbMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis ptpbMore data for this Ligand-Target Pair
Affinity DataIC50: 9.28E+3nMAssay Description:Inhibition of human leukocyte elastase using MeOSuc-Ala-Ala-Pro-Val-para-nitroanilide chromogenic substrate after 10 mins spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes without GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.47E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes with GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes with GTPMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human leukocyte elastase using MeOSuc-Ala-Ala-Pro-Val-para-nitroanilide chromogenic substrate after 10 mins spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranes without GTPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.83E+4nMAssay Description:Inhibition of human recombinant aromataseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of electric eel AChEMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Carica papaya papainMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Carica papaya papainMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Carica papaya papainMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Induction of NAD(P)H:quinone reductase in mouse Hepa 1c1c7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Induction of NAD(P)H:quinone reductase in mouse Hepa 1c1c7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Induction of NAD(P)H:quinone reductase in mouse Hepa 1c1c7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Induction of NAD(P)H:quinone reductase in mouse Hepa 1c1c7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human thrombinMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: 6.42E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis ptpbMore data for this Ligand-Target Pair
Affinity DataIC50: 6.56E+4nMAssay Description:Inhibition of forskolin-stimulated cAMP accumulation in chinese hamster ovary cell membranes expressing human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of forskolin-stimulated cAMP accumulation in chinese hamster ovary cell membranes expressing human adenosine A3 receptorMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHRMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDC25aMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTP1bMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDC25aMore data for this Ligand-Target Pair
TargetLow molecular weight protein-tyrosine phosphatase A(Mycobacterium tuberculosis)
University Of Bonn
Curated by ChEMBL
University Of Bonn
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis ptpAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDC25aMore data for this Ligand-Target Pair