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Found 93 with Last Name = 'karibe' and Initial = 'n'
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9410(N-[2-(1-benzylpiperidin-4-yl)ethyl]-N-ethyl-4-(phe...)
Affinity DataIC50:  0.300nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9409(CHEMBL299708 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)
Affinity DataIC50:  0.560nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9409(CHEMBL299708 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)
Affinity DataIC50:  0.600nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9411(CHEMBL54058 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  0.600nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004000((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...)
Affinity DataIC50:  0.690nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004016(CHEMBL138107 | CHEMBL544159 | N-(2-(2-(1-benzylpip...)
Affinity DataIC50:  1.20nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004007(2-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-1,3-dioxo-2,...)
Affinity DataIC50:  2.20nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004001(5-Benzoyl-2-[2-(1-benzyl-piperidin-4-yl)-ethyl]-is...)
Affinity DataIC50:  2.40nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004035(CHEMBL433678 | N-(2-(2-(1-benzylpiperidin-4-yl)eth...)
Affinity DataIC50:  2.80nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004018(3-(2-(1-benzylpiperidin-4-yl)ethyl)quinazoline-2,4...)
Affinity DataIC50:  4.20nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50003999(3-(2-(1-benzylpiperidin-4-yl)ethyl)-7-chloroquinaz...)
Affinity DataIC50:  4.5nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50003996(CHEMBL126354 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  5.40nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004011(2-(2-(1-benzylpiperidin-4-yl)ethyl)-5-methoxyisoin...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Rattus norvegicus (rat))
Eisai

Curated by ChEMBL
LigandPNGBDBM50004000((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...)
Affinity DataIC50:  8.10nMAssay Description:In vitro inhibitory concentration of the compound against butyrylcholinesterase (BuChE) obtained from rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50003998(5-Amino-2-[2-(1-benzyl-piperidin-4-yl)-ethyl]-isoi...)
Affinity DataIC50:  8.80nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004009(2-(2-(1-benzylpiperidin-4-yl)ethyl)-4-nitroisoindo...)
Affinity DataIC50:  9nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004015(4-Amino-2-[2-(1-benzyl-piperidin-4-yl)-ethyl]-isoi...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004040(2-(2-(1-benzylpiperidin-4-yl)ethyl)-5-nitroisoindo...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004033(3-(2-(1-benzylpiperidin-4-yl)ethyl)-3,4-dihydroqui...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004013(6-(2-(1-benzylpiperidin-4-yl)ethyl)-5H-pyrrolo[3,4...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004026(2-(2-(1-benzylpiperidin-4-yl)ethyl)-1,2-dihydroiso...)
Affinity DataIC50:  17nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004037(CHEMBL140737 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004012(2-(2-(1-benzylpiperidin-4-yl)ethyl)isoquinoline-1,...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9397(CHEMBL59583 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  29nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004020(2-(2-(1-benzylpiperidin-4-yl)ethyl)isoindoline-1,3...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9408((2E)-but-2-enedioic acid; N-[2-(1-benzylpiperidin-...)
Affinity DataIC50:  35nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9408((2E)-but-2-enedioic acid; N-[2-(1-benzylpiperidin-...)
Affinity DataIC50:  35nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9400((2E)-but-2-enedioic acid; N-[2-(1-benzylpiperidin-...)
Affinity DataIC50:  39nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004017(CHEMBL127527 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  46nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9396(CHEMBL56001 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  51nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004027(CHEMBL340672 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  52nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9391(N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-nitrobenzami...)
Affinity DataIC50:  55nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004036(CHEMBL340621 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  64nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004028(CHEMBL141167 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  65nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9399(CHEMBL299313 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)
Affinity DataIC50:  69nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Rattus norvegicus (rat))
Eisai

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  73nMAssay Description:In vitro inhibitory concentration of the compound against Butyrylcholinesterase obtained from rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  81nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9395(CHEMBL56706 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  85nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9392(CHEMBL54835 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  88nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004022(2-(2-(1-benzylpiperidin-4-yl)ethyl)isoindolin-1-on...)
Affinity DataIC50:  98nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004030(CHEMBL141352 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  108nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9393(CHEMBL56586 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  120nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9406(CHEMBL57696 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  130nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9413(CHEMBL127750 | N-methyl-N-(2-{1-[(3-methylphenyl)m...)
Affinity DataIC50:  145nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9401(4-{[2-(1-benzylpiperidin-4-yl)ethyl]carbamoyl}-1-o...)
Affinity DataIC50:  155nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9405(CHEMBL56470 | N-[2-(1-Benzyl-piperidin-4-yl)-ethyl...)
Affinity DataIC50:  170nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9405(CHEMBL56470 | N-[2-(1-Benzyl-piperidin-4-yl)-ethyl...)
Affinity DataIC50:  170nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9388(N-[2-(1-benzylpiperidin-4-yl)ethyl]-4-methylbenzam...)
Affinity DataIC50:  180nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM9394(CHEMBL55253 | N-[2-(1-benzylpiperidin-4-yl)ethyl]-...)
Affinity DataIC50:  180nMpH: 7.4 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
Tsukuba Research Laboratories

LigandPNGBDBM50004002(CHEMBL340609 | N-(2-(1-benzylpiperidin-4-yl)ethyl)...)
Affinity DataIC50:  205nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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