Affinity DataKi: 1.10nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 148nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 166nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 174nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 177nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 178nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 407nMAssay Description:Displacement of [3H]valsartan from human AT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of [3H]valsartan from human AT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Compound was evaluated for affinity towards human tachykinin NK-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 631nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 831nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 1.32E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 2.14E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.45E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.45E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.95E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.46E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.57E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 5.37E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.37E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.49E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.49E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 5.75E+3nMAssay Description:Inhibition of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.88E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.58E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.33E+3nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.46E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.91E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: <9.99E+4nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.70E+5nMAssay Description:Inhibition of human recombinant APN expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human recombinant DNMT1 expressed in H19 cells assessed as inhibition of tritiated methyl incorporation from [3H]-labeled AdoMet into h...More data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human recombinant DNMT1 expressed in H19 cells assessed as inhibition of tritiated methyl incorporation from [3H]-labeled AdoMet into h...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant DNMT1 expressed in H19 cells assessed as inhibition of tritiated methyl incorporation from [3H]-labeled AdoMet into h...More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of human recombinant DNMT1 expressed in H19 cells assessed as inhibition of tritiated methyl incorporation from [3H]-labeled AdoMet into h...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human recombinant DNMT1 expressed in H19 cells assessed as inhibition of tritiated methyl incorporation from [3H]-labeled AdoMet into h...More data for this Ligand-Target Pair