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Found 189 with Last Name = 'karpoormath' and Initial = 'r'
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232182(CHEMBL4097327)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50087713((1-Ethyl-propyl)-[3-(4-methoxy-2-methyl-phenyl)-2,...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I-Tyr0]-CRF from recombinant human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232188(CHEMBL4070141)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232179(CHEMBL4105538)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I-Tyr0]-CRF from recombinant human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232182(CHEMBL4097327)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232178(CHEMBL4081285)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I-Tyr0]-CRF from recombinant human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50116095(CHEMBL293228 | [3-(2,4-Dichloro-phenyl)-2,5-dimeth...)
Affinity DataKi:  2nMAssay Description:Displacement of 125I-sauvagine from CRF1 receptor in human IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50116123(Butyl-[3-(2,4-dichloro-phenyl)-2,5-dimethyl-2H-pyr...)
Affinity DataKi:  2nMAssay Description:Displacement of 125I-sauvagine from CRF1 receptor in human IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232191(CHEMBL4089611)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232188(CHEMBL4070141)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232191(CHEMBL4089611)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232201(CHEMBL4099753)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50116093(CHEMBL304335 | [3-(2,4-Dichloro-phenyl)-2,5-dimeth...)
Affinity DataKi:  3nMAssay Description:Displacement of 125I-sauvagine from CRF1 receptor in human IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50116118(CHEMBL304272 | [3-(2,4-Dichloro-phenyl)-2,5-dimeth...)
Affinity DataKi:  3nMAssay Description:Displacement of 125I-sauvagine from CRF1 receptor in human IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232190(CHEMBL4061482)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]Ro5-4864 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232201(CHEMBL4099753)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232190(CHEMBL4061482)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]PK11195 from PBZR in rat kidney mitochondrial membranes measured after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232183(CHEMBL4097805)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]o-CRF from recombinant human CRF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232200(CHEMBL4081736)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha1 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha5 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha1 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3(Rattus norvegicus)
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha3 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha2 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha1 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha2 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3(Rattus norvegicus)
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi:  383nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha3 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232200(CHEMBL4081736)
Affinity DataKi:  740nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha5 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM50232200(CHEMBL4081736)
Affinity DataKi:  927nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha2 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123830(4,5-dibromo-N'-(4-chlorobenzylidene)-1-methyl-...)
Affinity DataKi:  2.10E+3nM ΔG°:  -33.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123825(4,5-dibromo-N'-[(4-fluorophenyl)methylidene]-1...)
Affinity DataKi:  2.40E+3nM ΔG°:  -33.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123833(4,5-dibromo-N'-(2,4-dichlorobenzylidene)-1-met...)
Affinity DataKi:  2.60E+3nM ΔG°:  -33.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123832(4,5-dibromo-N'-(4-methoxybenzylidene)-1-methyl...)
Affinity DataKi:  2.90E+3nM ΔG°:  -32.9kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123823(4,5-dibromo-N'-[(2,4-dichlorophenyl)methyliden...)
Affinity DataKi:  3.10E+3nM ΔG°:  -32.7kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123831(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1-me...)
Affinity DataKi:  3.40E+3nM ΔG°:  -32.5kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123820(4,5-dibromo-N'-[(4-chlorophenyl)methylidene]-1...)
Affinity DataKi:  3.90E+3nM ΔG°:  -32.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123828(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1-met...)
Affinity DataKi:  3.90E+3nM ΔG°:  -32.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123824(4,5-dibromo-N'-(2-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  4.70E+3nM ΔG°:  -31.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123815(4,5-dibromo-N'-(4-fluorobenzylidene)-1H-pyrrol...)
Affinity DataKi:  5.10E+3nM ΔG°:  -31.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123818(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1Hpyr...)
Affinity DataKi:  5.20E+3nM ΔG°:  -31.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123829(4,5-dibromo-N'-(3,4-dihydroxybenzylidene)-1-me...)
Affinity DataKi:  6.10E+3nM ΔG°:  -31.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123822(4,5-dibromo-N'-(4-methoxybenzylidene)-1Hpyrrol...)
Affinity DataKi:  6.55E+3nM ΔG°:  -30.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123826(4,5-dibromo-1-methyl-N'-(4-nitrobenzylidene)-1...)
Affinity DataKi:  6.90E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123827(4,5-dibromo-N'-(4-hydroxybenzylidene)-1-methyl...)
Affinity DataKi:  7.10E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123814(4,5-dibromo-N'-(2-hydroxybenzylidene)-1H-pyrro...)
Affinity DataKi:  8.90E+3nM ΔG°:  -30.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123823(4,5-dibromo-N'-[(2,4-dichlorophenyl)methyliden...)
Affinity DataKi:  9.40E+3nM ΔG°:  -29.8kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]RO15-1788 from recombinant rat GABAalpha5 receptor expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123821(4,5-dibromo-N'-(3,4-dimethoxybenzylidene)-1Hpy...)
Affinity DataKi:  1.13E+4nM ΔG°:  -29.4kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123828(4,5-dibromo-N'-(2,6-dichlorobenzylidene)-1-met...)
Affinity DataKi:  1.23E+4nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123820(4,5-dibromo-N'-[(4-chlorophenyl)methylidene]-1...)
Affinity DataKi:  1.25E+4nM ΔG°:  -29.1kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Kwazulu-Natal

LigandPNGBDBM123833(4,5-dibromo-N'-(2,4-dichlorobenzylidene)-1-met...)
Affinity DataKi:  1.29E+4nM ΔG°:  -29.0kJ/molepH: 7.4 T: 2°CAssay Description:The reaction mixtures (200 uL), containing recombinant human MAO-A or MAO-B (5 ug/mL) and the test compounds in potassium phosphate buffer (100 mM; p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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