Found 1522 with Last Name = 'kim' and Initial = 'sy' 
Affinity DataKi: 0.160nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 0.610nM ΔG°: -54.7kJ/mole EC50: 12.2nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 0.920nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 1.83nM ΔG°: -51.9kJ/mole EC50: 5.20nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 3.29nM ΔG°: -50.4kJ/mole EC50: 12.1nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 3.40nMAssay Description:Antagonist activity for rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 3.40nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 3.60nM ΔG°: -50.1kJ/mole EC50: 12.3nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University
Seoul National University
Affinity DataKi: 4.12nM ΔG°: -49.8kJ/mole EC50: 0.580nMpH: 7.4 T: 2°CAssay Description:Binding assay mixtures were set up and contained [3H] RTX, various concentrations of competing ligands, and rVR1-transfected CHO cells. Nonspecific b...More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Research Institute Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:The inhibitory activity of the enteropeptidase inhibitor synthesized using the purified Recombinant Human Enteropeptidase and the substrate Acetyl-As...More data for this Ligand-Target Pair
