Affinity DataKi: 0.190nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity against Adenosine A1 receptor from rat forebrain membranes with N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.990nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity against Adenosine A2 receptor of striatal membrane using [3H]CGS-21680More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor of rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 1.73nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor of rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity for Adenosine A2 receptor using N-[3H]-ethyladenosine-5`-uronamide in presence of cyclopentyladenosine rat striatal membranes under ...More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity at Adenosine A2 receptor from rat striatal membranes by N-[3H] ethyladenosin-5'- uronamide displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity against Adenosine A2 receptor of striatal membrane using [3H]CGS-21680More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against Adenosine A1 receptor from rat forebrain membranes with N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of human factor 10a by Dixon-plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro binding affinity against Adenosine A2a receptor in rat forebrain membranes by [3H]-NECA (+CPA) displacement.More data for this Ligand-Target Pair