Affinity DataKi: 0.0530nMAssay Description:Inhibitory constant against bovine spleen Adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Inhibitory constant against bovine spleen Adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Inhibitory constant against bovine spleen Adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in pig cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.311nMAssay Description:Displacement of [3H]-CCPA from human recombinant adenosine A1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.313nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.345nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.386nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.387nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.393nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.429nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.432nMAssay Description:Displacement of [3H]-CCPA from human recombinant adenosine A1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.438nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.453nMAssay Description:Displacement of [3H]-CCPA from human recombinant adenosine A1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.454nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.461nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Inhibitory constant against bovine spleen Adenosine deaminaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.478nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptors was determined in bovine cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in pig cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.532nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.538nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.575nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.588nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Inhibition of [3H]- U-69593 binding in cloned rat Opioid receptor kappa 1 expressed in CHO cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 0.682nMAssay Description:Displacement of [3H]-CCPA from human recombinant adenosine A1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.728nMAssay Description:Displacement of [3H]-CCPA from human recombinant adenosine A1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]DAMGO from recombinant human mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.768nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity for human adenosine A1 receptor subtype expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.806nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.864nMAssay Description:Displacement of [3H]CCPA from recombinant human adenosine A1 receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.875nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Inhibition of [3H]U-69593 binding to Opioid receptor kappa 1 in guinea pig brain homogenatesMore data for this Ligand-Target Pair