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Found 102 with Last Name = 'lee' and Initial = 'jt'
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440172(CHEMBL2426574)
Affinity DataKi:  0.5nMAssay Description:Inhibition of dCK (unknown origin) by steady-state kinetic assayMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440173(CHEMBL2426573)
Affinity DataKi:  0.800nMAssay Description:Inhibition of dCK (unknown origin) by steady-state kinetic assayMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440151(CHEMBL2426558)
Affinity DataKi:  1.5nMAssay Description:Inhibition of dCK (unknown origin) by steady-state kinetic assayMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440140(CHEMBL2426588)
Affinity DataKi:  9.5nMAssay Description:Inhibition of dCK (unknown origin) by steady-state kinetic assayMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440183(CHEMBL2426563)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440176(CHEMBL2426570)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440173(CHEMBL2426573)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440177(CHEMBL2426569)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440184(CHEMBL2426562)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440179(CHEMBL2426567)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440182(CHEMBL2426564)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440174(CHEMBL2426572)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440175(CHEMBL2426571)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440151(CHEMBL2426558)
Affinity DataIC50:  3nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440151(CHEMBL2426558)
Affinity DataIC50:  3nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440172(CHEMBL2426574)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440155(CHEMBL2426598)
Affinity DataIC50:  7nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440180(CHEMBL2426566)
Affinity DataIC50:  8nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440152(CHEMBL2426557)
Affinity DataIC50:  11nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440181(CHEMBL2426565)
Affinity DataIC50:  12nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf [V600E](Homo sapiens (Human))
Plexxikon

LigandPNGBDBM25617(N-[3-({5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl}carb...)
Affinity DataIC50:  13nMpH: 7.0 T: 2°CAssay Description:The in vitro kinase activities of wild type or mutants were determined by measuring phosphorylation of biotinylated-MEK protein using Perkin-Elmer s ...More data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440140(CHEMBL2426588)
Affinity DataIC50:  18nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440178(CHEMBL2426568)
Affinity DataIC50:  19nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440155(CHEMBL2426598)
Affinity DataIC50:  30nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440148(CHEMBL2426561)
Affinity DataIC50:  31nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440140(CHEMBL2426588)
Affinity DataIC50:  35nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440149(CHEMBL2426560)
Affinity DataIC50:  37nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440153(CHEMBL2426460)
Affinity DataIC50:  83nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440162(CHEMBL2426591)
Affinity DataIC50:  92nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Plexxikon

LigandPNGBDBM25617(N-[3-({5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl}carb...)
Affinity DataIC50:  130nMpH: 7.5 T: 2°CAssay Description:Enzyme activity was assayed using Z-LYTE Enzymatic Kinase Assay format (Invitrogen Corp., Carlsbad, CA) according to the manufacturer instructions.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440164(CHEMBL2426589)
Affinity DataIC50:  150nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Plexxikon

LigandPNGBDBM25617(N-[3-({5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl}carb...)
Affinity DataIC50:  160nMpH: 7.0 T: 2°CAssay Description:The in vitro kinase activities of wild type or mutants were determined by measuring phosphorylation of biotinylated-MEK protein using Perkin-Elmer s ...More data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440154(CHEMBL2426459)
Affinity DataIC50:  162nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440149(CHEMBL2426560)
Affinity DataIC50:  170nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440150(CHEMBL2426559)
Affinity DataIC50:  173nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440148(CHEMBL2426561)
Affinity DataIC50:  175nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440143(CHEMBL2426585)
Affinity DataIC50:  197nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440146(CHEMBL2426582)
Affinity DataIC50:  230nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440163(CHEMBL2426590)
Affinity DataIC50:  230nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440145(CHEMBL2426583)
Affinity DataIC50:  251nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440162(CHEMBL2426591)
Affinity DataIC50:  255nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440153(CHEMBL2426460)
Affinity DataIC50:  265nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440157(CHEMBL2426596)
Affinity DataIC50:  297nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440143(CHEMBL2426585)
Affinity DataIC50:  330nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440150(CHEMBL2426559)
Affinity DataIC50:  385nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440163(CHEMBL2426590)
Affinity DataIC50:  395nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440147(CHEMBL2426581)
Affinity DataIC50:  421nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440160(CHEMBL2426593)
Affinity DataIC50:  506nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Mus musculus)
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440152(CHEMBL2426557)
Affinity DataIC50:  510nMAssay Description:Inhibition of dCK in mouse L1210 cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDeoxycytidine kinase(Homo sapiens (Human))
California Nanosystems Institute

Curated by ChEMBL
LigandPNGBDBM50440159(CHEMBL2426594)
Affinity DataIC50:  512nMAssay Description:Inhibition of dCK in human CCRF-CEM cells assessed as inhibition of tritiated deoxycytidine [3H]-dC uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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