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Found 46 with Last Name = 'lin' and Initial = 'ts'
TargetCytidine deaminase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50087289(1-beta-D-Arabinofuranosylcytosine | 4-Amino-1-beta...)
Affinity DataKi:  1.90E+5nMAssay Description:Inhibitory constant was measured on cytidine/deoxycytidine deaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCytidine deaminase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50007155(4-Amino-1-(3-hydroxy-5-hydroxymethyl-4-methylene-t...)
Affinity DataKi:  1.60E+6nMAssay Description:Inhibitory constant was measured on cytidine/deoxycytidine deaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytidine deaminase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50421893(CHEMBL10128)
Affinity DataKi:  7.69E+6nMAssay Description:Inhibitory constant was measured on cytidine/deoxycytidine deaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytidine deaminase(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50007156(4-Amino-5-fluoro-1-(4-hydroxy-5-hydroxymethyl-3-me...)
Affinity DataKi:  2.51E+7nMAssay Description:Inhibitory constant was measured on cytidine/deoxycytidine deaminaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051772((Z)-N'-(5-amino-6-formylpyridin-2-yl)carbamohydraz...)
Affinity DataIC50:  820nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051768((1Z,N'E)-N'-((3-(methylamino)pyridin-2-yl)methylen...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051776((1Z,N'E)-N'-((5-(ethylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051769((1Z,N'E)-N'-((5-(methylamino)pyridin-2-yl)methylen...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051775((1Z,N'E)-N'-((5-(allylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051767((1Z,N'E)-N'-((5-(propylamino)pyridin-2-yl)methylen...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051774((1Z,N'E)-N'-((3-(allylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051766((1Z,N'E)-N'-((5-(butylamino)pyridin-2-yl)methylene...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051777((1Z,N'E)-N'-((5-(aminomethyl)pyridin-2-yl)methylen...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051773((Z)-N'-(3-amino-6-formylpyridin-2-yl)carbamohydraz...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051771((1Z,N'E)-N'-((3,5-diaminopyridin-2-yl)methylene)ca...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonucleoside-diphosphate reductase subunit M2(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50051770((1Z,N'E)-N'-((5-amino-4-(morpholinomethyl)pyridin-...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory activity against CDP reductase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442476(CHEMBL2440365)
Affinity DataEC50:  3.40E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442486(CHEMBL2440381)
Affinity DataEC50:  3.30E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442487(CHEMBL2440370)
Affinity DataEC50:  2.90E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442488(CHEMBL2440374)
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442488(CHEMBL2440374)
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442472(CHEMBL2440369)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442475(CHEMBL2440366)
Affinity DataEC50:  1.10E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442477(CHEMBL2440378)
Affinity DataEC50:  5.10E+3nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442478(CHEMBL2440376)
Affinity DataEC50:  3.70E+3nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442474(CHEMBL2440367)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442487(CHEMBL2440370)
Affinity DataEC50:  620nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM20875(1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihyd...)
Affinity DataEC50:  120nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM20875(1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihyd...)
Affinity DataEC50:  77nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442479(CHEMBL2440371)
Affinity DataEC50:  3.50E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442473(CHEMBL2440368)
Affinity DataEC50:  4.60E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442486(CHEMBL2440381)
Affinity DataEC50:  4.70E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442485(CHEMBL2440372)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442484(CHEMBL2440373)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442483(CHEMBL2440375)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442482(CHEMBL2440377)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442481(CHEMBL2440379)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442480(CHEMBL2440380)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442478(CHEMBL2440376)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442477(CHEMBL2440378)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442476(CHEMBL2440365)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442475(CHEMBL2440366)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442474(CHEMBL2440367)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442473(CHEMBL2440368)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442472(CHEMBL2440369)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50442479(CHEMBL2440371)
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells assessed as inhibition of [14C]-AMG uptake up to 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed